SCHEMBL30141452

SCHEMBL30141452

CC(Oc1ccc2[nH]ncc2c1)c1cc(F)cc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.42
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
MAOB P27338 1/20 0.41
RAB9A P51151 5/20 0.40
NPC1 O15118 4/20 0.40
ROCK1 Q13464 4/20 0.40
NOS1 P29475 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CSNK2A1 P68400 2/20 0.40
METAP2 P50579 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TRPA1 O75762 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16023025 0.79 RAB9A (0.50) ROCK2MAOBRAB9ANPC1ROCK1
SCHEMBL5417396 0.78 ESR1 (0.44) ROCK2MAOBRAB9ANPC1ROCK1
SCHEMBL5408031 0.78 MEN1 (0.42) ROCK2MAOBRAB9ANPC1ROCK1
SCHEMBL28707122 0.77 NOS1 (0.46) ROCK2CTNNB1WNT3AMAOBRAB9A
SCHEMBL23622136 0.77 NR3C1 (0.47) ROCK2
SCHEMBL14738568 0.76 MAPT (0.52) ROCK2CTNNB1WNT3AMAOBRAB9A
SCHEMBL30540770 0.76 KDR (0.56) NOS1FGFR1FGFR2
SCHEMBL30498934 0.76 KDR (0.56) NOS1FGFR1FGFR2
SCHEMBL1336326 0.75 JAK2 (0.41) ROCK2ROCK1CSNK2A1FGFR1FGFR2
SCHEMBL23622250 0.74 NR3C1 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268080-A1 TRK KINASE INHIBITOR COMPOUND AND USE THEREOF 河南迈英诺医药科技有限公司 2022-12-29 WO disclosed