SCHEMBL301469

SCHEMBL301469

c1ccc(-c2ncco2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.71
LTA4H P09960 2/20 0.69
HDAC4 P56524 1/20 0.50
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NOTUM Q6P988 2/20 0.45
ATAD2 Q6PL18 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 1/20 0.42
BRD4 O60885 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
CASP1 P29466 1/20 0.42
CHRNA7 P36544 1/20 0.41
CHRNA10 Q9GZZ6 1/20 0.41
CHRNA9 Q9UGM1 1/20 0.41
PIN1 Q13526 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28753616 0.98 HPGDS (0.69) HPGDSLTA4HHDAC4NPC1RAB9A
SCHEMBL5571760 0.96 LTA4H (0.70) HPGDSLTA4HHDAC4NPC1RAB9A
Toluene SCHEMBL28904988 0.90 HPGDS (0.61) HPGDSLTA4HHDAC4NPC1RAB9A
Thiophene SCHEMBL19467814 0.88 HPGDS (0.59) HPGDSLTA4HHDAC4NPC1RAB9A
Acetic Acid SCHEMBL27259016 0.88 HPGDS (0.59) HPGDSLTA4HHDAC4NPC1RAB9A
SCHEMBL7979723 0.88 HPGDS (0.59) HPGDSLTA4HHDAC4NPC1RAB9A
Alcohol SCHEMBL27719231 0.88 HPGDS (0.59) HPGDSLTA4HHDAC4NPC1RAB9A
Piperazine SCHEMBL3360835 0.88 HPGDS (0.59) HPGDSLTA4HHDAC4NPC1RAB9A
Perchlorate SCHEMBL9472619 0.88 HPGDS (0.59) HPGDSLTA4HHDAC4NPC1RAB9A
SCHEMBL722557 0.87 LTA4H (0.64) HPGDSLTA4HHDAC4NOTUMBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2509 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119143678-A Fluorescent molecule for rapidly measuring excitation light spot size and light intensity distribution and preparation method thereof 中国科学院化学研究所 2024-12-17 CN claimed
US-20240026127-A1 COMPOSITE PARTICLE AND USE THEREOF IN OPTICAL FILTRATION COLOURSMITH LABS INC. (CA) 2024-01-25 US claimed
EP-4255983-A1 COMPOSITE PARTICLE AND USE THEREOF IN OPTICAL FILTRATION Coloursmith Labs Inc. (CA) 2023-10-11 EP claimed
US-20230197540-A1 ELECTRICAL TRACES ON GLASS CORES IN INTEGRATED CIRCUIT PACKAGES AND METHODS OF MANUFACTURING THE SAME INTEL CORPORATION 2023-06-22 US claimed
US-20230158025-A1 GALACTOKINASE INHIBITORS NATIONAL INSTITUTES OF HEALTH 2023-05-25 US claimed
CN-113896902-B Synthetic method and application of Ni (II) -based metal organic framework material 三峡大学 2022-09-16 CN claimed
WO-2022115948-A1 COMPOSITE PARTICLE AND USE THEREOF IN OPTICAL FILTRATION COLOURSMITH LABS INC. (CA) 2022-06-09 WO claimed
EP-2652810-B9 METHOD OF FORMING A RADIATION-EMITTING ORGANIC-ELECTRONIC DEVICE OSRAM OLED GMBH (DE) 2021-11-10 EP claimed
WO-2021216812-A1 GALACTOKINASE INHIBITORS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2021-10-28 WO claimed
EP-2652810-B1 METHOD OF FORMING A RADIATION-EMITTING ORGANIC-ELECTRONIC DEVICE OSRAM OLED GMBH (DE) 2021-08-11 EP claimed
EP-0733216-B1 A METHOD AND MATERIAL FOR THE DETECTION OF IONISING RADIATION BRITISH NUCLEAR FUELS PLC (GB) 2000-01-19 EP claimed
WO-1999008130-A1 METHOD AND DEVICE FOR RADIOGRAPHIC IMAGING USING GAMMA RAYS AND X-RAY BEAMS BIO - SCAN S.A. (CH) 1999-02-18 WO claimed
CN-1181720-A Remotely programmable matrices with memories and uses thereof IRORI (US) 1998-05-13 CN claimed
EP-0471756-A4 SACCHARIN DERIVATIVES USEFUL AS PROTEOLYTIC ENZYME INHIBITORS AND PREPARATION THEREOF 1992-04-08 EP claimed
EP-0471756-A1 SACCHARIN DERIVATIVES USEFUL AS PROTEOLYTIC ENZYME INHIBITORS AND PREPARATION THEREOF. STERLING WINTHROP INC (US) 1992-02-26 EP claimed
EP-0281012-B1 4-CHLORO-OXAZOLE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1991-12-11 EP claimed
WO-1990013549-A1 SACCHARIN DERIVATIVES USEFUL AS PROTEOLYTIC ENZYME INHIBITORS AND PREPARATION THEREOF STERLING WINTHROP INC. (US) 1990-11-15 WO claimed
US-4892799-A PHOTOCONDUCTIVITY, ELECTROGRAPHY HOECHST AKTIENGESELLSCHAFT (DE) 1990-01-09 US claimed
EP-0281012-A1 4-Chloro-oxazole derivatives, method for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1988-09-07 EP claimed
US-4067804-A POLYOXADIAZOLE RESIN THE FURUKAWA ELECTRIC COMPANY, LIMITED (JA) 1978-01-10 US claimed