SCHEMBL30149804

SCHEMBL30149804

Cc1ccc(S(=O)(=O)NN=C(c2cccnc2)C2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
STS P08842 5/20 0.48
MMP13 P45452 1/20 0.48
KMT2A Q03164 2/20 0.48
GPR119 Q8TDV5 4/20 0.47
CCNA2 P20248 1/20 0.46
CDK2 P24941 1/20 0.46
EGFR P00533 1/20 0.45
PTGS2 P35354 1/20 0.45
NAMPT P43490 1/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 1/20 0.44
MEN1 O00255 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SFRP1 Q8N474 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23211955 1.00 STS (0.48) STSMMP13KMT2AGPR119CCNA2
SCHEMBL23211953 1.00 STS (0.48) STSMMP13KMT2AGPR119CCNA2
SCHEMBL23211969 0.89 STS (0.52) STSMMP13KMT2AGPR119NAMPT
SCHEMBL23211970 0.89 STS (0.52) STSMMP13KMT2AGPR119NAMPT
SCHEMBL22773317 0.89 MMP13 (0.55) STSMMP13KMT2AGPR119MEN1
SCHEMBL22773318 0.89 MMP13 (0.55) STSMMP13KMT2AGPR119MEN1
SCHEMBL25260321 0.89 MMP13 (0.55) STSMMP13KMT2AGPR119MEN1
SCHEMBL21382156 0.87 EGFR (0.50) KMT2AEGFRPTGS2NAMPTLMNA
SCHEMBL21382157 0.87 EGFR (0.50) KMT2AEGFRPTGS2NAMPTLMNA
SCHEMBL22491580 0.84 KMT2A (0.53) STSMMP13KMT2AGPR119MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230117324-A1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2023-04-20 US disclosed
EP-3768684-B1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS HOFFMANN LA ROCHE (CH) 2023-02-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230117324-A1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS MGLL, LPL, LIPC STS 388/4885MMP13 663/4885KMT2A 2681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.