SCHEMBL3015286

SCHEMBL3015286

NC(=O)c1ccc(O)c(N)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.55
PARP1 P09874 2/20 0.54
GAA P10253 5/20 0.47
MAPT P10636 3/20 0.47
CA2 P00918 2/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA9 Q16790 1/20 0.47
ALDH1A1 P00352 7/20 0.46
HSD17B10 Q99714 5/20 0.46
ALOX15 P16050 3/20 0.46
ALOX12 P18054 3/20 0.46
HPGD P15428 2/20 0.46
MAPK1 P28482 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 2/20 0.46
ERN1 O75460 2/20 0.46
THRB P10828 1/20 0.44
TSHR P16473 1/20 0.42
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336990 0.84 ALDH1A1 (0.53) GAAMAPTCA2CA12CA1
SCHEMBL30786420 0.84 ALDH1A1 (0.53) GAAMAPTCA2CA12CA1
SCHEMBL79989 0.82 KDM4E (0.64) GAAMAPTCA2CA12CA1
SCHEMBL5595306 0.82 LCK (0.55) LCKPARP1GAAMAPTCA2
SCHEMBL29476052 0.82 KDM4E (0.64) GAAMAPTCA2CA12CA1
Protocatechuamide SCHEMBL1128716 0.81 LCK (0.65) LCKPARP1GAAMAPTCA2
SCHEMBL1428434 0.81 ALDH1A1 (0.49) LCKPARP1MAPTALDH1A1HSD17B10
SCHEMBL8412857 0.81 ALDH1A1 (0.49) LCKPARP1MAPTALDH1A1HSD17B10
SCHEMBL9307729 0.80 KDM4E (0.61) GAAMAPTCA2CA12CA1
SCHEMBL3287715 0.80 PRKCI (0.58) GAAMAPTCA2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103288757-B Preparation method of 6-amino-7-hydroxyl-3,4-dihydroquinazoline-4-ketone SUZHOU MINGRUI PHARMACEUTICAL TECHNOLOGY CO LTD 2015-07-01 CN claimed
CN-103265497-B Intermediate compound 4-chloro-6-amino-7-hydroxyquinazoline required for synthesis of tinib antineoplastic drug and preparation method thereof SUZHOU MIRACPHARMA TECHNOLOGY CO LTD 2014-11-26 CN claimed
CN-103288757-A Preparation method of 6-amino-7-hydroxyl-3,4-dihydroquinazoline-4-ketone SUZHOU MINGRUI PHARMACEUTICAL TECHNOLOGY CO LTD 2013-09-11 CN claimed
CN-103265497-A Intermediate compound 4-chloro-6-amino-7-hydroxyquinazoline required for synthesis of tinib antineoplastic drug and preparation method thereof SUZHOU MINGYUE MEDICAL TECHNOLOGY CO LTD 2013-08-28 CN claimed
EP-3383854-B1 WATER-SOLUBLE UV-ABSORBING COMPOUNDS AND USES THEREOF ALCON INC (CH) 2021-03-03 EP disclosed
US-10301598-B2 Low-molecular-compound for improving production, maintenance and proliferation of pluripotent stem cells, composition comprising the same, and culture method KOREA RESEARCH INSTITUTE OF BIOSCIENCE AND BIOTECHNOLOGY (KR) 2019-05-28 US disclosed
US-20170159023-A1 NOVEL LOW-MOLECULAR-COMPOUND FOR IMPROVING PRODUCTION, MAINTENANCE AND PROLIFERATION OF PLURIPOTENT STEM CELLS, COMPOSITION COMPRISING THE SAME, AND CULTURE METHOD KOREA RESEARCH INSTITUTE OF BIOSCIENCE AND BIOTECHNOLOGY (KR) 2017-06-08 US disclosed
WO-2017093835-A1 WATER-SOLUBLE UV-ABSORBING COMPOUNDS AND USES THEREOF NOVARTIS AG (CH) 2017-06-08 WO disclosed
EP-2774918-B1 NOVEL LOW-MOLECULAR WEIGHT COMPOUND FOR PROMOTING PLURIPOTENT STEM CELL GENERATION, MAINTENANCE, AND PROLIFERATION, AND COMPOSITION AND CULTURING METHOD CONTAINING SAME KOREA RES INST BIOSCIENCE & BIOTECHNOLOGY (KR) 2017-03-22 EP disclosed
US-9587225-B2 Low-molecular-compound for improving production, maintenance and proliferation of pluripotent stem cells, composition comprising the same, and culture method KOREA RESEARCH INSTITUTE OF BIOSCIENCE AND BIOTECHNOLOGY (KR) 2017-03-07 US disclosed
CN-103288757-B Preparation method of 6-amino-7-hydroxyl-3,4-dihydroquinazoline-4-ketone SUZHOU MINGRUI PHARMACEUTICAL TECHNOLOGY CO LTD 2015-07-01 CN disclosed
US-20150159142-A1 NOVEL LOW-MOLECULAR-COMPOUND FOR IMPROVING PRODUCTION, MAINTENANCE AND PROLIFERATION OF PLURIPOTENT STEM CELLS, COMPOSITION COMPRISING THE SAME, AND CULTURE METHOD Korea Reasearch Institute of Bioscience and Biotechnology (KR) 2015-06-11 US disclosed
US-4563409-A ELECTROGRAPHY HOGOHAYA CHEMICAL CO., LTD. (JP) 1986-01-07 US disclosed
EP-0141377-A2 Metal complexes HODOGAYA CHEMICAL CO., LTD. (JP) 1985-05-15 EP disclosed
US-4141890-A FIBER-REACTIVE CIBA-GEIGY CORPORATION (US) 1979-02-27 US disclosed
US-RE29585-E DYEING WOOL CIBA-GEIGY CORPORATION (US) 1978-03-21 US disclosed
US-4067864-A FOR CELLULOSE OR POLYAMIDES CIBA-GEIGY AG (CH) 1978-01-10 US disclosed
US-4039523-A YELLOW CIBA-GEIGY AG (CH) 1977-08-02 US disclosed
US-4017477-A 3-Halogeno-6-hydroxy-pyridone-(2) azo dyestuffs CIBA-GEIGY AG (CH) 1977-04-12 US disclosed
US-3971738-A Heavy metal complexes of azo compounds containing a halogeno-2,3-dihydroxy pyridine coupling component CIBA-GEIGY AG (CH) 1976-07-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150159142-A1 NOVEL LOW-MOLECULAR-COMPOUND FOR IMPROVING PRODUCTION, MAINTENANCE AND PROLIFERATION OF PLURIPOTENT STEM CELLS, COMPOSITION COMPRISING THE SAME, AND CULTURE METHOD MYC, MYCBP, HES1 LCK 4610/4885PARP1 1057/4885GAA 4180/4885
US-10301598-B2 Low-molecular-compound for improving production, maintenance and proliferation of pluripotent stem cells, composition comprising the same, and culture method AANAT, MKI67, VIM LCK 4565/4885PARP1 385/4885GAA 4495/4885
US-20170159023-A1 NOVEL LOW-MOLECULAR-COMPOUND FOR IMPROVING PRODUCTION, MAINTENANCE AND PROLIFERATION OF PLURIPOTENT STEM CELLS, COMPOSITION COMPRISING THE SAME, AND CULTURE METHOD AANAT, MKI67, ACP1 LCK 4597/4885PARP1 658/4885GAA 4400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.