SCHEMBL30159547

SCHEMBL30159547

O=Cc1c(F)cc(Cl)cc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C4 P17516 1/20 0.44
AKR1C3 P42330 1/20 0.44
AKR1C2 P52895 1/20 0.44
AKR1C1 Q04828 1/20 0.44
CYP3A4 P08684 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ACLY P53396 5/20 0.38
DYRK1A Q13627 1/20 0.38
NOTUM Q6P988 1/20 0.38
TPMT P51580 1/20 0.38
TSHR P16473 1/20 0.37
CASP1 P29466 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23529330 1.00 AKR1C4 (0.44) AKR1C4AKR1C3AKR1C2AKR1C1CYP3A4
SCHEMBL23529377 0.81 ERN1 (0.47) AKR1C2AKR1C1CYP3A4KEAP1NFE2L2
SCHEMBL29948173 0.81 ERN1 (0.47) AKR1C2AKR1C1CYP3A4KEAP1NFE2L2
SCHEMBL906303 0.81 AKR1C4 (0.57) AKR1C4AKR1C3AKR1C2AKR1C1CYP3A4
SCHEMBL1349783 0.80 ERN1 (0.41) CYP3A4ALDH1A1HSD17B10TSHRGRM2
SCHEMBL11179328 0.75 ERN1 (0.43) CYP3A4ALDH1A1HPGDHSD17B10CA1
SCHEMBL23529333 0.75 ALDH1A1 (0.48) AKR1C4AKR1C3AKR1C2AKR1C1CYP3A4
SCHEMBL6242355 0.75 AKR1C2 (0.64) AKR1C4AKR1C3AKR1C2AKR1C1CYP3A4
SCHEMBL25296415 0.74 TSHR (0.41) CYP3A4KEAP1NFE2L2ALDH1A1TP53
SCHEMBL5357933 0.74 KEAP1 (0.46) AKR1C4AKR1C3AKR1C2AKR1C1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022266711-A1 SUBSTITUTED AMIDOBENZIMIDAZOLE DIMERS AS STING MODULATORS Aculeus Therapeutics Pty Ltd (AU) 2022-12-29 WO disclosed