SCHEMBL30165101

SCHEMBL30165101

[2H]c1ncc(C(F)(F)F)cc1F

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.37
CYP11B2 P19099 4/20 0.37
GPR55 Q9Y2T6 1/20 0.32
KIF11 P52732 1/20 0.31
IDH1 O75874 1/20 0.31
DAO P14920 1/20 0.31
CYP19A1 P11511 4/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.30
METAP2 P50579 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
SLC22A6 Q4U2R8 1/20 0.30
SLC22A8 Q8TCC7 1/20 0.30
SLC22A12 Q96S37 1/20 0.30
SLC22A11 Q9NSA0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690255 0.79 CYP11B1 (0.44) CYP11B1CYP11B2GPR55KIF11IDH1
SCHEMBL31305866 0.74
SCHEMBL3749196 0.73 CYP11B1 (0.43) CYP11B1CYP11B2KIF11DAOCYP19A1
SCHEMBL30803919 0.72 DAO (0.37) CYP11B1CYP11B2DAO
Piperazine SCHEMBL28793735 0.69 CHRNB2 (0.38) CYP11B1CYP11B2IDH1DAOALDH1A1
SCHEMBL30164989 0.69 KIF11 (0.37) CYP11B1CYP11B2KIF11CYP19A1ALDH1A1
SCHEMBL29791400 0.68 CYP19A1 (0.44) KIF11CYP19A1CYP1A2METAP2CYP3A4
SCHEMBL21744244 0.67 CYP11B2 (0.56) CYP11B1CYP11B2GPR55KIF11IDH1
SCHEMBL9693899 0.65 CES2 (0.42) ALDH1A1CYP3A4
SCHEMBL4461544 0.65 CES2 (0.48) ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006013-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2023-02-02 WO disclosed