SCHEMBL30165670

SCHEMBL30165670

O=C1COCCN1c1cccc(Br)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 2/20 0.43
ALOX5 P09917 2/20 0.43
PTGS2 P35354 10/20 0.43
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
JAK2 O60674 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30165667 1.00 MAP4K1 (0.43) MAP4K1ALOX5PTGS2CYP3A4CYP2D6
SCHEMBL19994364 1.00 MAP4K1 (0.43) MAP4K1ALOX5PTGS2CYP3A4CYP2D6
SCHEMBL25676559 0.78 MAP4K1 (0.46) MAP4K1PTGS2CYP3A4CYP2D6CYP2C9
SCHEMBL31334702 0.78 MAP4K1 (0.41) MAP4K1PTGS2CYP3A4CYP2D6CYP2C9
SCHEMBL4780 0.78 ALOX5 (0.46) MAP4K1ALOX5GRIN2DGRIN3BGRIN1
SCHEMBL3297331 0.77 PTGS2 (0.43) MAP4K1PTGS2CYP3A4CYP2D6CYP2C9
SCHEMBL29464219 0.76 PARP1 (0.48) MAP4K1ALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL19994372 0.76 PARP1 (0.48) MAP4K1ALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL31334775 0.75 PARP1 (0.47) MAP4K1ALOX5CYP3A4CYP2D6CYP2C9
SCHEMBL19994341 0.75 PARP1 (0.47) MAP4K1ALOX5CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110402248-B Azaindoles as HPK1 inhibitors 豪夫迈·罗氏有限公司 2023-01-06 CN disclosed