SCHEMBL30168076

SCHEMBL30168076

[C-]#[N+]c1ccccc1-n1ccc2ccc(C)cc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
CYP2A6 P11509 3/20 0.35
DOT1L Q8TEK3 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
HSP90AA1 P07900 1/20 0.34
MAOB P27338 1/20 0.33
P2RX7 Q99572 1/20 0.33
PRMT5 O14744 1/20 0.33
CYP19A1 P11511 1/20 0.32
HTR7 P34969 1/20 0.32
MAPT P10636 2/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP1A2 P05177 2/20 0.31
ROCK1 Q13464 1/20 0.31
MEN1 O00255 1/20 0.31
NR1I2 O75469 1/20 0.31
AHR P35869 1/20 0.31
KMT2A Q03164 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30168080 0.88 MAOB (0.44) HTR2AHTR2CCYP2A6TDP1HSP90AA1
SCHEMBL28893986 0.78 HTR2A (0.39) HTR2AHTR2CCYP2A6DOT1LTDP1
SCHEMBL30168069 0.76 MEN1 (0.35) CYP2A6TDP1P2RX7CYP1A2MEN1
SCHEMBL30168073 0.75 KCNH2 (0.38) HTR2AHTR2CCYP2A6HSP90AA1P2RX7
SCHEMBL29599854 0.75 BIRC5 (0.41) HTR2AHTR2CCYP2A6HSP90AA1PRMT5
SCHEMBL5661673 0.74 FGFR1 (0.47) HTR2AHTR2CCYP2A6TDP1MAOB
SCHEMBL29600322 0.73 HTR2A (0.37) HTR2AHTR2CCYP2A6P2RX7PRMT5
SCHEMBL22649105 0.71 TP53 (0.46) CYP2A6TDP1HSP90AA1MAOBMAPT
SCHEMBL6840186 0.71 RXRA (0.48) HSP90AA1ROCK1RAPGEF4
SCHEMBL13183604 0.70 HTR2A (0.45) HTR2AHTR2CCYP2A6TDP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115536662-A Guanyl structure-containing tetracyclic indole compound, and synthesis method and application thereof 广州大学 2022-12-30 CN disclosed