SCHEMBL30170784

SCHEMBL30170784

CN(C(=O)OC(C)(C)C)c1cc2ccccc2c(Br)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.43
BRD4 O60885 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.38
NCEH1 Q6PIU2 5/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GAA P10253 1/20 0.36
GBA1 P04062 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 3/20 0.34
KDM4E B2RXH2 2/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20315161 1.00 PAX8 (0.43) PAX8BRD4TRPM8NCEH1MEN1
SCHEMBL29517495 1.00 PAX8 (0.43) PAX8BRD4TRPM8NCEH1MEN1
SCHEMBL20296577 0.88 TRPM8 (0.38) PAX8BRD4TRPM8NCEH1MEN1
SCHEMBL20296817 0.80 MEN1 (0.43) TRPM8NCEH1MEN1KMT2AALDH1A1
SCHEMBL22029263 0.80 CTSS (0.37) PAX8TRPM8MEN1KMT2ANPC1
SCHEMBL3633134 0.77 PAX8 (0.43) PAX8BRD4TRPM8NCEH1ALDH1A1
SCHEMBL31453184 0.75 PAX8 (0.38) PAX8BRD4
SCHEMBL68085 0.75 PAX8 (0.42) PAX8BRD4NCEH1MEN1KMT2A
SCHEMBL4154983 0.74 TRPM8 (0.41) TRPM8MEN1KMT2AGAAALDH1A1
SCHEMBL17559731 0.73 MEN1 (0.44) TRPM8MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115626923-A KRAS G12C inhibitors and methods of use thereof 美国安进公司 2023-01-20 CN disclosed
CN-110997668-B KRAS G12C inhibitors and methods of use thereof 美国安进公司 2022-11-01 CN disclosed