SCHEMBL30178331

SCHEMBL30178331

COc1ccc(N)c(CCNC2CCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
EPHX2 P34913 1/20 0.53
STS P08842 2/20 0.49
MAPT P10636 3/20 0.46
TP53 P04637 1/20 0.46
BACE1 P56817 2/20 0.46
CTSD P07339 1/20 0.46
CTSE P14091 1/20 0.46
TGFBR1 P36897 2/20 0.45
HTT P42858 2/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
GPR119 Q8TDV5 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
DYRK1A Q13627 1/20 0.44
NPC1 O15118 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3651872 0.88 ALDH1A1 (0.56) ALDH1A1EPHX2STSMAPTTP53
SCHEMBL6517994 0.87 EPHX2 (0.46) ALDH1A1EPHX2STSMAPTTP53
SCHEMBL17870707 0.86 DRD4 (0.42) ALDH1A1EPHX2
SCHEMBL30178438 0.85 GPR119 (0.49) ALDH1A1EPHX2MAPTHTTCA12
SCHEMBL6520126 0.85 EPHX2 (0.47) ALDH1A1EPHX2STSMAPTTP53
SCHEMBL1814017 0.84 KDM4E (0.48) ALDH1A1STSMAPTHTTGPR119
SCHEMBL4321000 0.82 ALDH1A1 (0.52) ALDH1A1EPHX2STSMAPTTP53
SCHEMBL3652370 0.82 ALDH1A1 (0.52) ALDH1A1EPHX2STSMAPTTP53
SCHEMBL3652372 0.82 ALDH1A1 (0.52) ALDH1A1EPHX2STSMAPTTP53
SCHEMBL19873971 0.81 SIGMAR1 (0.41) EPHX2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3708566-B1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RES & DEV (FR) 2023-02-08 EP disclosed