SCHEMBL30182736

SCHEMBL30182736

O=C(O)c1ccc(C(=O)Nc2cnc(C3=CCNCC3)cn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.44
CCNT1 O60563 2/20 0.39
CDK9 P50750 2/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39
HDAC4 P56524 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
BRAF P15056 1/20 0.38
WNT3A P56704 2/20 0.38
P2RY14 Q15391 1/20 0.36
DEGS1 O15121 1/20 0.36
BTK Q06187 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
TSHR P16473 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24892328 0.83 MAPKAPK2 (0.43) WNT3AMAPKAPK2
SCHEMBL29803411 0.83 CCNT1 (0.49) CCNT1CDK9HDAC4HDAC6BRAF
SCHEMBL171560 0.79 P4HA1 (0.54) WNT3AP2RY14SIGMAR1GABRPGABRD
SCHEMBL24891691 0.77 DYRK1A (0.48) HCAR3WNT3ATSHR
SCHEMBL4746022 0.72 QDPR (0.62) P2RY14SIGMAR1GABRPGABRDGABRA1
SCHEMBL24891690 0.71 GRM1 (0.49) WNT3A
SCHEMBL24892089 0.71 WNT3A (0.43) CCNT1CDK9WNT3ATSHRMAPKAPK2
SCHEMBL30182219 0.71 WNT3A (0.43) CCNT1CDK9WNT3ATSHRMAPKAPK2
SCHEMBL24891851 0.71 WNT3A (0.43) WNT3ATSHRMAPKAPK2
SCHEMBL5225955 0.70 HDAC1 (0.51) HDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023287736-A1 NOVEL BIS-AMIDE CONTAINING COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2023-01-19 WO disclosed