SCHEMBL30189946

SCHEMBL30189946

CC(C)(O)COc1cc(N)ccn1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 4/20 0.45
ACACB O00763 1/20 0.38
IL1B P01584 1/20 0.37
LOX P28300 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
ASIC3 Q9UHC3 1/20 0.34
ACVR2A P27037 1/20 0.33
TGFBR2 P37173 1/20 0.33
AAK1 Q2M2I8 5/20 0.33
MCHR1 Q99705 1/20 0.33
PTGS2 P35354 2/20 0.33
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21379706 1.00 NUDT1 (0.45) NUDT1ACACBIL1BLOXLOXL2
SCHEMBL19783211 0.83 CYP2D6 (0.41) NUDT1LOXLOXL2ASIC3ACVR2A
SCHEMBL30189896 0.81 ALDH1A1 (0.41) NUDT1ACACBIL1BLOXLOXL2
SCHEMBL18150999 0.81 ALDH1A1 (0.41) NUDT1ACACBIL1BLOXLOXL2
SCHEMBL109903 0.80 ALDH1A1 (0.48) NUDT1LOXLOXL2ASIC3NOS3
SCHEMBL15464119 0.78 IL1B (0.49) IL1BMCHR1PTGS2NOS3NOS2
SCHEMBL28941077 0.77 MEN1 (0.41) NUDT1ACACBIL1BLOXL2AAK1
SCHEMBL2144434 0.76 LOXL2 (0.43) LOXLOXL2ASIC3NOS3NOS1
SCHEMBL2228010 0.75 KDM4E (0.49) NUDT1IL1B
SCHEMBL171947 0.75 TP53 (0.48) ACACBLOXLOXL2ASIC3NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed