SCHEMBL30197384

SCHEMBL30197384

Cc1cc(-c2ccc(F)cc2)ncc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.42
IDO1 P14902 1/20 0.42
NPC1 O15118 4/20 0.40
RXFP1 Q9HBX9 1/20 0.40
MAPK14 Q16539 2/20 0.39
AURKA O14965 1/20 0.39
ABL1 P00519 1/20 0.39
NTRK1 P04629 1/20 0.39
LCK P06239 1/20 0.39
CSF1R P07333 1/20 0.39
RET P07949 1/20 0.39
MET P08581 1/20 0.39
PDGFRB P09619 1/20 0.39
PIM1 P11309 1/20 0.39
PDGFRA P16234 1/20 0.39
FLT3 P36888 1/20 0.39
MAPK8 P45983 1/20 0.39
CDK8 P49336 1/20 0.39
MAP2K1 Q02750 1/20 0.39
MAP4K2 Q12851 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290369 1.00 TDO2 (0.42) TDO2IDO1NPC1RXFP1MAPK14
SCHEMBL27157143 0.85 LDHA (0.41) NPC1ABL1RETAURKBLDHA
SCHEMBL30819263 0.85 LDHA (0.41) NPC1ABL1RETAURKBLDHA
SCHEMBL31735547 0.84 GRM5 (0.39) METPIM1LDHAGRM5CYP1A2
SCHEMBL25755553 0.83 TDO2 (0.45) TDO2IDO1NPC1RXFP1MAPK14
SCHEMBL18015262 0.82 CYP1A2 (0.40) NPC1LDHARAB9AALDH1A1KDM4E
SCHEMBL15420845 0.81 LDHA (0.57) TDO2IDO1NPC1PDGFRBFLT3
SCHEMBL18015452 0.79 LDHA (0.41) TDO2IDO1NPC1MAPK14LDHA
SCHEMBL25752509 0.78 GAA (0.44) GRM5ALDH1A1KDM4EL3MBTL1GAA
SCHEMBL25752504 0.78 KMO (0.43) NPC1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed