SCHEMBL302050

SCHEMBL302050

O=S(=O)(c1cccnc1)N(Cc1ccc(Cl)cc1)c1cccc(N2CCOCC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.53
CNR2 P34972 4/20 0.52
PKM P14618 1/20 0.47
HTR1A P08908 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
HTR6 P50406 1/20 0.45
PLOD2 O00469 1/20 0.44
PLOD3 O60568 1/20 0.44
PLOD1 Q02809 1/20 0.44
EP300 Q09472 1/20 0.42
HIF1A Q16665 1/20 0.42
NAMPT P43490 2/20 0.41
CYP3A4 P08684 1/20 0.41
CNR1 P21554 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPC1 O15118 1/20 0.40
PTGER2 P43116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL302891 0.85 HTR2C (0.66) HTR2CCNR2HTR1AHTR2AHTR7
SCHEMBL302209 0.83 CNR2 (0.51) HTR2CCNR2PKMHTR1AHTR2A
SCHEMBL302085 0.81 CNR2 (0.47) HTR2CCNR2PKMHTR1AHTR2A
SCHEMBL301830 0.81 HTR2C (0.61) HTR2CCNR2PKMHTR1AHTR2A
SCHEMBL1976235 0.78 CNR2 (0.44) HTR2CCNR2HTR1AHTR2AHTR7
SCHEMBL303319 0.77 LMNA (0.48) CNR2PKMCYP3A4HTTPTGER2
SCHEMBL11401740 0.77 CNR2 (0.50) HTR2CCNR2PKMPLOD2PLOD3
SCHEMBL13064496 0.77 LMNA (0.58) CNR2PKMCYP3A4HTTSMN1; SMN2
SCHEMBL2246857 0.77 MEN1 (0.65) CNR2PKMCNR1HTTSMN1; SMN2
SCHEMBL1966404 0.76 DRD4 (0.51) HTR2CCNR2HTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500835-A 2012-01-12 JP claimed
EP-2334637-A1 NOVEL POTASSIUM CHANNEL BLOCKERS Xention Limited (GB) 2011-06-22 EP claimed