SCHEMBL302066

SCHEMBL302066

CN1C(=O)N(C)C(=O)C(O)(C2(O)C(=O)N(C)C(=O)N(C)C2=O)C1=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HPGD P15428 1/20 0.41
BLM P54132 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
ADRA2C P18825 1/20 0.30
GSK3A P49840 1/20 0.30
GSK3B P49841 1/20 0.30
MGLL Q99685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8609384 0.80 ALDH1A1 (0.40) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL10195453 0.73 LMNA (0.40) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL23733143 0.70 LMNA (0.34) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL2601688 0.69
SCHEMBL16091680 0.69 ALDH1A1 (0.34) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL23733068 0.69 ALDH1A1 (0.35) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL16091679 0.69 LMNA (0.37) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL12107403 0.67 LMNA (0.39) LMNAADRA2CGSK3AGSK3BMGLL
SCHEMBL11730000 0.67 ATM (0.50) ALDH1A1KDM4ELMNAL3MBTL1
SCHEMBL23733175 0.66 KDM4E (0.33) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120213855-A1 DOSAGE FORMS FOR WEAKLY IONIZABLE COMPOUNDS CIMA LABS INC. (US) 2012-08-23 US claimed
JP-2012500643-A 2012-01-12 JP claimed
US-20110223251-A1 BACTERIAL COMPOSITION CHR-HANSEN A/S 2011-09-15 US claimed
EP-2334302-A2 DOSAGE FORMS FOR WEAKLY IONIZABLE COMPOUNDS Cima Labs Inc. (US) 2011-06-22 EP claimed
EP-2318511-A1 BACTERIAL COMPOSITION Chr. Hansen A/S (DK) 2011-05-11 EP claimed
CN-101141949-B New pharmaceutical compositions useful in the treatment of parkinson's disease OREXO AB 2010-12-08 CN claimed
WO-2010030667-A2 DOSAGE FORMS FOR WEAKLY IONIZABLE COMPOUNDS CIMA LABS INC. (US) 2010-03-18 WO claimed
WO-2010023248-A1 Bacterial Composition CHR. HANSEN A/S (DK) 2010-03-04 WO claimed
US-20080193526-A1 Pharmaceutical Compositions Useful in the Treatment of Pain OREXO AB (SE) 2008-08-14 US claimed
CN-101141949-A New pharmaceutical compositions useful in the treatment of parkinson's disease OREXO AB (SE) 2008-03-12 CN claimed
EP-1863455-A1 NEW PHARMACEUTICAL COMPOSITIONS USEFUL IN THE TREATMENT OF PARKINSON'S DISEASE Orexo AB (SE) 2007-12-12 EP claimed
WO-2006103417-A1 NEW PHARMACEUTICAL COMPOSITIONS USEFUL IN THE TREATMENT OF PARKINSON'S DISEASE OREXO AB (SE) 2006-10-05 WO claimed
WO-2006078241-A1 EFFERVESCENT AND EFFERVESCENT-DISPERSION COMPOSITIONS FOR MEDICAMENTS AND METHODS OF USE THEREOF SERENE MEDICAL, INC. (US) 2006-07-27 WO claimed
US-20050074489-A1 Effervescent and effervescent-dispersion compositions for medicaments and methods of use thereof PEDIAMED PHARMACEUTICALS, INC. 2005-04-07 US claimed
US-20050031677-A1 Sequential drug delivery systems CIMA LABS INC. (US) 2005-02-10 US claimed
US-20030232080-A1 Sequential drug delivery systems CIMA LABS INC. (US) 2003-12-18 US claimed
CN-110590485-B FSO 2 N 3 Use in the production of azido compounds 中宏鑫投资控股(深圳)有限公司 2023-04-14 CN disclosed
CN-111417398-A Glycan formulations for treating infections 卡莱多生物科技有限公司 2020-07-14 CN disclosed
CN-1151117-A Binding of E-selectin, P-selectin or L-selectin to sialyl-Lewis(x) or sialyl-lewis(a) TAXAS BIOTECHNOLOGY CORP (US) 1997-06-04 CN disclosed
US-5525576-A CARBOHYDRATES AND POLYHYDROXYCARBOXYLIC ACIDS OBTAINED BY THE OXIDATION OF A HULL-FREE PENTOSE-CONTAINING EXTRACT; ENHANCED ABSORPTION OF PLANT GROWTH REGULATORS, INSECTICIDES, FUNGICIDES AND PESTICIDES MEDINA-VEGA LUIS R (US) 1996-06-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120213855-A1 DOSAGE FORMS FOR WEAKLY IONIZABLE COMPOUNDS ABCB11, CEL, SLC7A5 ALDH1A1 2213/4885KDM4E 3774/4885SMN1; SMN2 3245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.