SCHEMBL30209643

SCHEMBL30209643

Cc1ccc2nc(C=CC(N)=O)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 2/20 0.52
KDM4E B2RXH2 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
NFKB1 P19838 1/20 0.50
RAB9A P51151 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
HDAC8 Q9BY41 4/20 0.49
HDAC6 Q9UBN7 4/20 0.49
HDAC2 Q92769 3/20 0.49
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC7 Q8WUI4 2/20 0.49
HDAC10 Q969S8 2/20 0.49
HDAC11 Q96DB2 2/20 0.49
HDAC9 Q9UKV0 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3532231 0.86 KDM4E (0.62) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL3532228 0.86 KDM4E (0.62) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL30209641 0.82 HDAC8 (0.71) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL3590241 0.82 HDAC1 (0.71) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL3590247 0.82 HDAC1 (0.71) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL30209650 0.82 BACE1 (0.47) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL30209652 0.82 HDAC6 (0.46) PFKFB3KDM4ESMN1; SMN2ALDH1A1HDAC8
SCHEMBL30209657 0.82 MAPT (0.52) PFKFB3KDM4ESMN1; SMN2ALDH1A1HDAC8
SCHEMBL29596601 0.82 RAB9A (0.67) PFKFB3KDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL30209665 0.78 HDAC6 (0.53) PFKFB3KDM4ESMN1; SMN2ALDH1A1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115745898-A Aromatic acrylamide-triazole compound, and preparation method and application thereof 许昌学院 2023-03-07 CN disclosed