SCHEMBL30216623

SCHEMBL30216623

O=C1CCCN1[C@H](c1ccc(Cl)cc1)c1ccc(F)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
CYP3A4 P08684 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
MDM2 Q00987 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SCN8A Q9UQD0 1/20 0.37
MGLL Q99685 1/20 0.36
TP53 P04637 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
MAPT P10636 1/20 0.35
GPX4 P36969 1/20 0.35
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
KAT2B Q92831 2/20 0.34
PIN1 Q13526 1/20 0.34
GAA P10253 1/20 0.34
CHRM2 P08172 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30216634 1.00 KMT2A (0.38) KMT2AMEN1CYP3A4CYP1A2CYP2C19
SCHEMBL30216630 0.86 MEN1 (0.35) KMT2AMEN1CYP3A4CYP1A2CYP2C19
SCHEMBL1002847 0.76 MCHR1 (0.36) KMT2AADRA1AADRA1BCHRM2CHRM4
SCHEMBL1004285 0.70 LMNA (0.40) CYP3A4ADRA1A
SCHEMBL7441149 0.69 HSD17B2 (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL3551369 0.69 LMNA (0.41) CYP3A4CYP2C19MDM2SMN1; SMN2MGLL
SCHEMBL5718440 0.67 CHRM2 (0.46) KMT2AMEN1CYP3A4CYP1A2CYP2C19
SCHEMBL3556189 0.67 MCHR1 (0.44) KMT2AADRA1AGAACHRM2CHRM4
SCHEMBL13074142 0.64 PER2 (0.39) KMT2AMEN1MAPTADRA1AADRA1B
SCHEMBL29915095 0.64 DRD2 (0.53) KMT2AMEN1CYP1A2CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115697327-A 5-oxo-pyrrolidine-3-carboxamides as NAV1.8 inhibitors 默沙东有限责任公司 2023-02-03 CN disclosed