SCHEMBL30296207

SCHEMBL30296207

CCCCc1nc(C)c(CC(=O)N(C)C)c(=O)[nH]1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.43
TSHR P16473 1/20 0.43
LMNA P02545 1/20 0.42
KDM4E B2RXH2 4/20 0.42
PARP1 P09874 1/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 2/20 0.40
THRB P10828 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26688859 0.85 LMNA (0.51) MAPK1TSHRLMNAKDM4EPARP1
SCHEMBL20778195 0.84 MAPK1 (0.63) MAPK1TSHRLMNAKDM4EPARP1
SCHEMBL1891525 0.81 TSHR (0.43) MAPK1TSHRLMNAKDM4EPARP1
SCHEMBL26688878 0.81 PKM (0.41) MAPK1TSHRLMNAKDM4EALDH1A1
SCHEMBL9490757 0.79 KDM4E (0.50) MAPK1TSHRLMNAKDM4EPARP1
SCHEMBL2227651 0.75 LMNA (0.39) TSHRLMNAKDM4EPOLBL3MBTL1
SCHEMBL25778574 0.75 KDM4E (0.55) LMNAKDM4EPARP1POLBL3MBTL1
SCHEMBL26688805 0.74 PKM (0.63) TSHRKDM4EALDH1A1THRBMEN1
SCHEMBL20778200 0.74 KDM4E (0.52) TSHRLMNAKDM4EPARP1L3MBTL1
SCHEMBL9487922 0.73 PARP1 (0.51) MAPK1KDM4EPARP1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117836294-A Biological antagonist containing aromatic ring, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-04-05 CN disclosed
WO-2023025277-A1 AROMATIC RING-CONTAINING BIOLOGICAL ANTAGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2023-03-02 WO disclosed