SCHEMBL30296246

SCHEMBL30296246

COCc1cncc(-c2cc(F)c(N)cc2Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.41
CYP11B1 P15538 5/20 0.41
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
TLR7 Q9NYK1 2/20 0.34
KCNH2 Q12809 4/20 0.34
GRIN2B Q13224 2/20 0.32
CYP2D6 P10635 1/20 0.32
PRMT6 Q96LA8 1/20 0.32
GRM5 P41594 2/20 0.32
TDO2 P48775 1/20 0.31
CYP17A1 P05093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26461083 0.83 CYP11B1 (0.32) CYP11B2CYP11B1PRMT6TDO2
SCHEMBL30296327 0.83 CYP11B1 (0.32) CYP11B2CYP11B1PRMT6TDO2
SCHEMBL31026729 0.80 CYP11B1 (0.46) CYP11B2CYP11B1CYP17A1
SCHEMBL26469046 0.77 CYP11B2 (0.43) CYP11B2CYP11B1TDO2CYP17A1
SCHEMBL30296491 0.77 CYP11B2 (0.43) CYP11B2CYP11B1TDO2CYP17A1
SCHEMBL30296367 0.75 PIK3CA (0.44) KCNH2
SCHEMBL30296489 0.74 CYP2A6 (0.50) CYP11B2CYP11B1
SCHEMBL30296737 0.73 EPHB4 (0.36) KCNH2GRIN2BTDO2
SCHEMBL30296309 0.72 CYP11B2 (0.42) CYP11B2CYP11B1PRMT5WDR77TLR7
SCHEMBL30296533 0.71 PIK3CA (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240368173-A1 TRICYCLIC GPR65 MODULATORS Pathios Therapeutics Limited (GB) 2024-11-07 US disclosed
EP-4419203-A1 TRICYCLIC GPR65 MODULATORS Pathios Therapeutics Limited (GB) 2024-08-28 EP disclosed
CN-118451080-A Tricyclic GPR65 modulators 帕蒂奥斯治疗有限公司 2024-08-06 CN disclosed
WO-2023067322-A1 TRICYCLIC GPR65 MODULATORS Pathios Therapeutics Limited (GB) 2023-04-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240368173-A1 TRICYCLIC GPR65 MODULATORS GPR65, GPR3, NR1H2 CYP11B2 328/4885CYP11B1 309/4885PRMT5 3110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.