SCHEMBL3029696

SCHEMBL3029696

CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CC(C)[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.67
SHBG P04278 6/20 0.67
CYP2C19 P33261 4/20 0.67
NR3C1 P04150 4/20 0.67
SERPINA6 P08185 3/20 0.67
MAPT P10636 3/20 0.67
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
SMN1; SMN2 Q16637 3/20 0.67
BLM P54132 2/20 0.67
ADORA3 P0DMS8 1/20 0.67
MAPK3 P27361 1/20 0.67
SLC6A3 Q01959 1/20 0.67
HIF1A Q16665 5/20 0.53
HSD17B10 Q99714 3/20 0.53
TSHR P16473 3/20 0.53
CYP3A4 P08684 2/20 0.53
PMP22 Q01453 1/20 0.53
PGR P06401 3/20 0.51
ALDH1A1 P00352 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3777671 0.89 LMNA (0.67) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL3777666 0.89 LMNA (0.67) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL10425177 0.88 HSD17B10 (0.69) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL28750427 0.88 LMNA (0.66) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL9705874 0.87 SHBG (0.66) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL9705867 0.87 SHBG (0.66) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL571164 0.85 LMNA (0.62) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL8415805 0.83 NR3C1 (0.56) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL8415802 0.83 NR3C1 (0.56) LMNASHBGCYP2C19NR3C1SERPINA6
SCHEMBL9643566 0.82 SHBG (0.48) LMNASHBGCYP2C19NR3C1SERPINA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8236791-B2 Assays for S100 inhibitors ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2012-08-07 US disclosed
US-20100216776-A1 Assays for S100 inhibitors ALBERT EINSTEIN COLLEGE OF MEDICINE 2010-08-26 US disclosed
WO-2008094410-A9 PARALLEL PROFILING OF SIGNALING PATHWAYS EINSTEIN COLL MED (US) 2008-10-02 WO disclosed
WO-2008094410-A2 PARALLEL PROFILING OF SIGNALING PATHWAYS ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2008-08-07 WO disclosed
WO-2008054354-A2 ASSAYS FOR S1OO INHIBITORS ALBERT EINSTEIN COLLEGE OF MEDECINE OF YESHIVA UNIVERSITY (US) 2008-05-08 WO disclosed