SCHEMBL30309564

SCHEMBL30309564

CS(=O)(=O)c1ccc(-c2cn3ccc(F)cc3n2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.65
SCD O00767 1/20 0.64
KDM4E B2RXH2 8/20 0.53
ALDH1A1 P00352 5/20 0.53
MEN1 O00255 1/20 0.53
HSP90AA1 P07900 1/20 0.53
KMT2A Q03164 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
NPC1 O15118 8/20 0.52
RAB9A P51151 8/20 0.52
MAPT P10636 2/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
TP53 P04637 2/20 0.50
GLA P06280 1/20 0.50
HPGD P15428 3/20 0.49
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
GFER P55789 1/20 0.48
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL913809 0.85 SCD (0.79) HDAC6SCDKDM4EALDH1A1MEN1
SCHEMBL30966874 0.85 SMN1; SMN2 (0.71) HDAC6SCDKDM4EALDH1A1MEN1
SCHEMBL915138 0.83 SCD (0.78) HDAC6SCDKDM4EALDH1A1MEN1
Zolimidine SCHEMBL932657 0.79 HDAC6 (1.00) HDAC6SCDKDM4EALDH1A1MEN1
SCHEMBL22615001 0.79 RAB9A (0.60) KDM4EALDH1A1MEN1KMT2ANPC1
SCHEMBL913165 0.78 SCD (0.76) HDAC6SCDKDM4EALDH1A1MEN1
SCHEMBL28909326 0.78 TLR9 (0.61) SCDKDM4EALDH1A1KMT2ANPC1
Zolimidine SCHEMBL29405502 0.78 HDAC6 (0.97) HDAC6SCDKDM4EALDH1A1MEN1
SCHEMBL914100 0.78 SCD (0.74) HDAC6SCDKDM4EALDH1A1MEN1
SCHEMBL14067368 0.75 TLR9 (0.48) SCDKDM4EALDH1A1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096717-A Imidazo [1,2-a ] pyridine and [1,2,4] triazolo [1,5-a ] pyridine derivatives as TLR9 inhibitors for the treatment of fibrosis 百时美施贵宝公司 2023-05-09 CN claimed
CN-116096717-A Imidazo [1,2-a ] pyridine and [1,2,4] triazolo [1,5-a ] pyridine derivatives as TLR9 inhibitors for the treatment of fibrosis 百时美施贵宝公司 2023-05-09 CN disclosed