SCHEMBL303115

SCHEMBL303115

Cc1ccccc1S(=O)(=O)N(Cc1ccccc1)c1ccc(C(=O)N2CCN(c3ccccc3)CC2)cc1.Cn1cnc(S(=O)(=O)N(Cc2ccccc2)c2ccc(C(=O)N3CCN(c4ccccc4)CC3)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
HTT P42858 1/20 0.52
GAA P10253 1/20 0.47
KMT2A Q03164 2/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.44
REV1 Q9UBZ9 1/20 0.43
OXTR P30559 1/20 0.42
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
FNTA P49354 2/20 0.41
FNTB P49356 2/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
PGGT1B P53609 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1722406 0.93 LMNA (0.58) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL1723243 0.90 LMNA (0.54) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL1711134 0.89 LMNA (0.63) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL1725046 0.86 LMNA (0.54) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL303692 0.86 LMNA (0.66) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL306227 0.85 TSHR (0.49) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL1725647 0.84 LMNA (0.53) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL3275527 0.83 LMNA (0.51) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL302045 0.82 SLC6A7 (0.53) LMNASMN1; SMN2HTTGAAKMT2A
SCHEMBL1723336 0.81 LMNA (0.57) LMNASMN1; SMN2HTTGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500834-A 2012-01-12 JP claimed
EP-2344456-A1 NOVEL POTASSIUM CHANNEL BLOCKER Xention Limited (GB) 2011-07-20 EP claimed
WO-2010023445-A1 NOVEL POTASSIUM CHANNEL BLOCKER XENTION LIMITED (GB) 2010-03-04 WO claimed