SCHEMBL30329263

SCHEMBL30329263

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1cnc(C(F)(F)F)cn1)C2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.48
RET P07949 7/20 0.46
GPR119 Q8TDV5 3/20 0.45
ACACB O00763 3/20 0.43
EIF2AK4 Q9P2K8 1/20 0.42
CYP2D6 P10635 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP1A2 P05177 2/20 0.41
TSHR P16473 2/20 0.41
CKS1B P61024 1/20 0.41
SKP1 P63208 1/20 0.41
SKP2 Q13309 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
CYP3A4 P08684 2/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30328476 0.93 GPR119 (0.49) CYP11B2RETGPR119CYP2D6HSD17B10
SCHEMBL30328958 0.90 CYP11B2 (0.46) CYP11B2RETGPR119ACACBEIF2AK4
SCHEMBL30898352 0.86 RET (0.43) CYP11B2RETGPR119EIF2AK4CKS1B
SCHEMBL30409946 0.86 RET (0.43) CYP11B2RETGPR119EIF2AK4CKS1B
SCHEMBL31296441 0.85 CKS1B (0.55) GPR119CKS1BSKP1SKP2HPGD
SCHEMBL21521592 0.85 CKS1B (0.55) GPR119CKS1BSKP1SKP2HPGD
SCHEMBL25164474 0.85 CYP11B2 (0.55) CYP11B2RETGPR119ACACBEIF2AK4
SCHEMBL30328050 0.85 CYP11B2 (0.55) CYP11B2RETGPR119ACACBEIF2AK4
SCHEMBL30327742 0.84 CYP11B2 (0.49) CYP11B2RETGPR119ACACBHSD17B10
SCHEMBL30327956 0.83 HDAC1 (0.39) CYP11B2GPR119ACACBCKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4415706-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-08-21 EP disclosed
WO-2023064343-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2023-04-20 WO disclosed