SCHEMBL3035294

SCHEMBL3035294

Cc1ccc(-c2ccccc2)n1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.88

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.88
ALDH1A1 P00352 3/20 0.61
MAPT P10636 2/20 0.61
PKM P14618 2/20 0.61
HTT P42858 1/20 0.61
PTGER1 P34995 3/20 0.58
ALOX5 P09917 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
KDM4E B2RXH2 1/20 0.56
HPGD P15428 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
PTGS1 P23219 2/20 0.54
MYC P01106 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6517559 0.97 PTGS2 (0.89) PTGS2ALDH1A1MAPTPKMHTT
SCHEMBL3831175 0.94 PTGS2 (1.00) PTGS2ALDH1A1MAPTPKMHTT
SCHEMBL7212097 0.88 PTGS2 (1.00) PTGS2ALDH1A1MAPTPTGER1KDM4E
SCHEMBL3021477 0.86 PTGS2 (0.67) PTGS2ALDH1A1MAPTPKMHTT
SCHEMBL6513769 0.85 PTGS2 (0.78) PTGS2ALDH1A1MAPTPTGER1KDM4E
SCHEMBL7215254 0.85 PTGS2 (0.78) PTGS2ALDH1A1MAPTPTGER1KDM4E
SCHEMBL5309102 0.85 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL7210644 0.85 PTGS2 (0.78) PTGS2ALDH1A1MAPTPKMHTT
SCHEMBL3026333 0.85 PTGS2 (0.78) PTGS2ALDH1A1MAPTPTGER1KDM4E
SCHEMBL3025180 0.84 PTGS2 (0.68) PTGS2ALDH1A1MAPTPKMHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8609713-B2 Pyrrole derivatives and their methods of use ABBVIE INC. (US) 2013-12-17 US disclosed
US-20100216748-A1 Pyrrole Derivatives and Their Methods of Use ABBOTT LABORATORIES (US) 2010-08-26 US disclosed
US-7741364-B2 Neuronal nicotinic acetylcholine receptor modulators; such as ethyl 1-[4-(aminosulfonyl)phenyl]-5-(4-bromophenyl)-2-methyl-1H-pyrrole-3-carboxylate ABBOTT LABORATORIES (US) 2010-06-22 US disclosed
CN-101479241-A Pyrrole derivatives and their methods of use ABBOTT LAB (US) 2009-07-08 CN disclosed
US-20080064695-A1 PYRROLE DERIVATIVES AND THEIR METHODS OF USE ABBVIE INC. 2008-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064695-A1 PYRROLE DERIVATIVES AND THEIR METHODS OF USE PYCR1, PPOX, DHPS PTGS2 69/4885ALDH1A1 745/4885MAPT 1215/4885
US-20100216748-A1 Pyrrole Derivatives and Their Methods of Use PYCR1, PPOX, DHPS PTGS2 69/4885ALDH1A1 745/4885MAPT 1215/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.