SCHEMBL30358449

SCHEMBL30358449

CNC(=O)C1CC(n2cnc3cccc(C(N)=O)c32)C1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.37
IDO1 P14902 3/20 0.37
KCNH2 Q12809 3/20 0.37
DPP4 P27487 2/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
PARP1 P09874 3/20 0.34
USP2 O75604 1/20 0.33
SYK P43405 4/20 0.33
RXFP1 Q9HBX9 1/20 0.33
JAK1 P23458 2/20 0.32
CYP11B2 P19099 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
ABL2 P42684 1/20 0.32
DPP8 Q6V1X1 1/20 0.31
PIK3C3 Q8NEB9 1/20 0.31
JAK3 P52333 1/20 0.31
BTK Q06187 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2507230 0.75 USP2 (0.41) CYP2C9IDO1KCNH2DRD2DRD3
SCHEMBL31030883 0.74 IDO1 (0.45) CYP2C9IDO1KCNH2
SCHEMBL27929032 0.70 DPP4 (0.58) DPP4PARP1SYKDPP8
SCHEMBL30121941 0.64 PARP1 (0.40) DPP4PARP1
SCHEMBL31196366 0.63 USP2 (0.49) CYP2C9IDO1KCNH2DRD2USP2
SCHEMBL24932847 0.62 DRD2 (0.38) CYP2C9IDO1KCNH2DPP4DRD2
SCHEMBL28284464 0.62 PIK3C3 (0.44) PARP1SYKPIK3C3BTK
SCHEMBL31196498 0.61 MKNK1 (0.47) CYP2C9IDO1KCNH2DRD2USP2
SCHEMBL31196386 0.61 MKNK1 (0.47) CYP2C9IDO1KCNH2DRD2USP2
SCHEMBL30843989 0.58 SLC9A1 (0.42) DPP4PARP1DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023004291-A1 CORONAVIRUS MAIN PROTEASE INHIBITORS AND METHODS USING SAME BAYLOR COLLEGE OF MEDICINE (US) 2023-01-26 WO disclosed