SCHEMBL30359155

SCHEMBL30359155

Cc1nc(C(=O)N2C3CCC2CNC3)c(C)o1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
TRPV4 Q9HBA0 1/20 0.34
MGLL Q99685 1/20 0.33
NAMPT P43490 1/20 0.33
CHRNA4 P43681 10/20 0.32
CHRNB2 P17787 3/20 0.31
CHRNB4 P30926 3/20 0.31
CHRNA3 P32297 3/20 0.31
CHRNA7 P36544 2/20 0.31
SPR P35270 1/20 0.30
HTR2C P28335 1/20 0.30
SSTR2 P30874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30358997 0.79 KCNK3 (0.41) KCNK3KCNK9TRPV4NAMPTCHRNA4
SCHEMBL30359148 0.75 CHRNA4 (0.43) KCNK3KCNK9TRPV4NAMPTCHRNA4
SCHEMBL30358999 0.70 KCNK3 (0.42) KCNK3KCNK9TRPV4NAMPTCHRNA4
SCHEMBL30359111 0.69 HTR2A (0.41) KCNK3KCNK9CHRNA4CHRNB2CHRNB4
SCHEMBL30359020 0.68 TRPV4 (0.40) KCNK3KCNK9TRPV4CHRNA4CHRNB2
SCHEMBL30359067 0.67 KCNK3 (0.45) KCNK3KCNK9TRPV4CHRNA4CHRNB2
SCHEMBL30359028 0.67 TRPV4 (0.41) TRPV4MGLLCHRNA4SPR
SCHEMBL30359106 0.66 KCNK3 (0.43) KCNK3KCNK9TRPV4CHRNA4CHRNB2
SCHEMBL30359077 0.64 ALDH1A1 (0.48) MGLL
SCHEMBL2302714 0.64 CHRNB2 (0.45) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed