SCHEMBL30361968

SCHEMBL30361968

N#Cc1ccc(F)c(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.51
XDH P47989 1/20 0.45
SLC22A12 Q96S37 1/20 0.45
GRM5 P41594 2/20 0.44
VNN1 O95497 1/20 0.44
HTT P42858 1/20 0.43
PIN1 Q13526 1/20 0.41
NOTUM Q6P988 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KAT6A Q92794 1/20 0.40
HSD17B14 Q9BPX1 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
P4HB P07237 1/20 0.40
TRPA1 O75762 1/20 0.40
ALB P02768 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL284291 1.00 MAP2K1 (0.51) MAP2K1XDHSLC22A12GRM5VNN1
SCHEMBL389029 0.85 MAP2K1 (0.55) MAP2K1XDHSLC22A12HTTMEN1
SCHEMBL29726442 0.83 CASP1 (0.44) MAP2K1GRM5VNN1HTTMEN1
SCHEMBL282483 0.83 ALDH1A1 (0.47) MAP2K1GRM5VNN1HTTMEN1
SCHEMBL923754 0.83 CASP1 (0.44) MAP2K1GRM5VNN1HTTMEN1
SCHEMBL7213897 0.83 GRM5 (0.46) MAP2K1GRM5VNN1MEN1KMT2A
SCHEMBL31494319 0.82 XDH (0.67) XDHSLC22A12HTTPIN1
SCHEMBL3157619 0.82 XDH (0.53) MAP2K1XDHSLC22A12HTTPIN1
SCHEMBL1477071 0.82 GRM5 (0.44) MAP2K1SLC22A12GRM5VNN1
SCHEMBL20564443 0.81 CYP3A4 (0.40) MAP2K1ALBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4665733-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 Bristol-Myers Squibb Company (US) 2025-12-24 EP disclosed
EP-4422746-A1 RXFP1 AGONISTS Bristol-Myers Squibb Company (US) 2024-09-04 EP disclosed
WO-2024173323-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 BRISTOL-MYERS SQUIBB COMPANY (US) 2024-08-22 WO disclosed
WO-2023076626-A1 RXFP1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-05-04 WO disclosed