Medazepam

Medazepam

SCHEMBL30366342

[2H]C1CN=C(c2ccccc2)c2cc(Cl)ccc2N1C

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 8/20 0.76
PDE4D Q08499 2/20 0.76
NR1I2 O75469 2/20 0.76
ADORA3 P0DMS8 2/20 0.76
HTR2C P28335 1/20 0.76
ADRA1A P35348 1/20 0.76
PTGS2 P35354 1/20 0.76
CHRNA4 P43681 1/20 0.76
SLC6A3 Q01959 1/20 0.76
GABRA1 P14867 2/20 0.58
GABRA5 P31644 2/20 0.58
GABRA3 P34903 2/20 0.58
GABRA2 P47869 2/20 0.58
GABRB2 P47870 2/20 0.58
GABRP O00591 1/20 0.58
GABRD O14764 1/20 0.58
CACNA1F O60840 1/20 0.58
ALB P02768 1/20 0.58
GABRB1 P18505 1/20 0.58
GABRG2 P18507 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Medazepam SCHEMBL11658148 0.86 OPRK1 (1.00) OPRK1PDE4DNR1I2ADORA3HTR2C
Medazepam SCHEMBL18472 0.86 OPRK1 (1.00) OPRK1PDE4DNR1I2ADORA3HTR2C
Medazepam SCHEMBL29642025 0.86 OPRK1 (1.00) OPRK1PDE4DNR1I2ADORA3HTR2C
Medazepam SCHEMBL78352 0.85 OPRK1 (0.97) OPRK1PDE4DNR1I2ADORA3HTR2C
SCHEMBL14018729 0.78 OPRK1 (0.84) OPRK1PDE4DNR1I2ADORA3HTR2C
SCHEMBL10917026 0.77 OPRK1 (0.65) OPRK1PDE4DNR1I2ADORA3HTR2C
SCHEMBL10917030 0.77 OPRK1 (0.65) OPRK1PDE4DNR1I2ADORA3HTR2C
SCHEMBL5692828 0.77 GABRA1 (0.77) OPRK1PDE4DNR1I2ADORA3HTR2C
SCHEMBL5692824 0.77 GABRA1 (0.77) OPRK1PDE4DNR1I2ADORA3HTR2C
Hydrochloric Acid SCHEMBL10922304 0.76 OPRK1 (0.64) OPRK1PDE4DNR1I2ADORA3HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111679002-B Kit for anxiolytic and hypnotic drugs in serum by ultra-high performance liquid chromatography tandem mass spectrometry technology 南京品生医疗科技有限公司 2023-05-09 CN disclosed