SCHEMBL30409441

SCHEMBL30409441

Cc1c(CN(C)C)c2ccc(C=O)cc2n1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.39
HDAC6 Q9UBN7 5/20 0.38
HDAC1 Q13547 4/20 0.38
HDAC2 Q92769 3/20 0.38
PTGER4 P35408 3/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 2/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRNA7 P36544 1/20 0.33
BRD4 O60885 1/20 0.33
BRD2 P25440 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
BRD7 Q9NPI1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL327664 0.78 CYP2A6 (0.53) CYP2A6PTGER4MAPTKMT2AALDH1A1
SCHEMBL30410104 0.77 ALDH1A1 (0.40) CYP2A6PTGER4MAPTKMT2AMAPK1
SCHEMBL30408484 0.77 CYP2A6 (0.46) CYP2A6PTGER4MAPTKMT2ANPC1
SCHEMBL30409974 0.76 ERN1 (0.44) MAPTKMT2ANPSR1ALDH1A1MEN1
SCHEMBL30409773 0.75 CNR1 (0.47) MAPTKMT2AALDH1A1MEN1GAA
SCHEMBL11180624 0.70 GPR3 (0.57) CYP2A6PTGER4MAPTKMT2ANPC1
SCHEMBL1911800 0.67 MAPT (0.53) CYP2A6PTGER4MAPTKMT2ANPC1
SCHEMBL18104492 0.66 PTGER4 (0.61) CYP2A6PTGER4MAPTKMT2AMAPK1
SCHEMBL18269303 0.66 PLA2G4A (0.46) HDAC6HDAC1HDAC2PTGER4MAPT
SCHEMBL18029372 0.65 USP14 (0.35) MAPTKMT2AMAPK1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116133658-A Novel compounds as inhibitors of histone deacetylase 6 and pharmaceutical compositions comprising the same 株式会社 钟根堂 2023-05-16 CN disclosed