SCHEMBL30414722

SCHEMBL30414722

NC(=O)c1ccnn1-c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.48
HTT P42858 1/20 0.45
MAP4K4 O95819 2/20 0.42
NPC1 O15118 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PTGS2 P35354 3/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA9 Q16790 1/20 0.40
F2 P00734 1/20 0.40
PLAU P00749 1/20 0.40
KLKB1 P03952 1/20 0.40
ELANE P08246 1/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL406516 0.86 ALDH1A1 (0.41) NR3C2HTTNPC1CYP1A2CYP2D6
SCHEMBL4951225 0.83 HSD17B10 (0.41) NR3C2NPC1RAB9AMEN1KMT2A
SCHEMBL3168308 0.82 POLB (0.53) NR3C2CYP2C19MEN1KMT2APOLB
SCHEMBL27134892 0.82 CCNC (0.42) NR3C2CYP1A2CYP2D6CYP2C19POLB
SCHEMBL28258620 0.82 NPBWR1 (0.40) PTGS1SMN1; SMN2
SCHEMBL15428737 0.82 NR3C2 (0.52) NR3C2HTTNPC1RAB9AMEN1
SCHEMBL10926946 0.81 XDH (0.46) HTTNPC1RAB9AMEN1KMT2A
SCHEMBL30853122 0.80 LMNA (0.36) CYP1A2CYP2C19KLKB1PARP1
SCHEMBL4953424 0.80 POLB (0.43) NR3C2NPC1CYP2C19RAB9APOLB
SCHEMBL15428570 0.78 HTT (0.45) NR3C2HTTRAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057646-B Pyrazole derivative and application thereof in preparation of antitumor drugs 常州大学 2023-05-02 CN disclosed