SCHEMBL30429201

SCHEMBL30429201

Cc1ccc(C#N)n1CCCCl

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.33
PGR P06401 3/20 0.32
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 3/20 0.31
MAPT P10636 3/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
AR P10275 6/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30429215 0.95 PGR (0.33) PRKCIPGRKDM4EALDH1A1MAPT
SCHEMBL28545999 0.81 PGR (0.46) PGRKDM4EALDH1A1MAPTMEN1
SCHEMBL19301845 0.71 AR (0.47) PGRKDM4EALDH1A1MAPTL3MBTL1
SCHEMBL31263971 0.68 DRD3 (0.36) KDM4EALDH1A1MAPTL3MBTL1MEN1
SCHEMBL19301847 0.68 SIGMAR1 (0.39) PGR
SCHEMBL2955486 0.68
SCHEMBL14859724 0.67 EPHX2 (0.36) ALDH1A1MEN1KMT2A
SCHEMBL22366341 0.67 AR (0.34) AR
SCHEMBL19301778 0.66 ALDH1A1 (0.56) KDM4EALDH1A1MAPTL3MBTL1MEN1
SCHEMBL19301772 0.65 GABRA1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111511750-B Macrocyclic derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2023-06-13 CN disclosed