SCHEMBL304342

SCHEMBL304342

CCOC(=O)C(Cc1ccc(C(N)=O)cc1)=C(C(=O)O)C(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 4/20 0.40
PLA2G10 O15496 1/20 0.38
PLA2G2A P14555 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
F2 P00734 3/20 0.37
F10 P00742 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HTT P42858 1/20 0.36
PLG P00747 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
C1S P09871 1/20 0.35
PRSS3 P35030 1/20 0.35
DPP4 P27487 2/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL304845 0.90 ALDH1A1 (0.42) MEN1KMT2AALDH1A1MAPT
SCHEMBL10193636 0.86 PLA2G10 (0.46) PARP10PLA2G10PLA2G2AF2PLG
SCHEMBL304961 0.85 CA2 (0.41) MEN1KMT2A
SCHEMBL305147 0.85 PLA2G10 (0.45) PARP10PLA2G10PLA2G2AF2PLG
SCHEMBL305149 0.85 PLA2G10 (0.45) PARP10PLA2G10PLA2G2AF2PLG
SCHEMBL304236 0.83 L3MBTL1 (0.38) ALDH1A1MAPT
SCHEMBL305321 0.82 KMT2A (0.38) MEN1KMT2AALDH1A1HTTMAPT
SCHEMBL305802 0.81 SMN1; SMN2 (0.32) MEN1KMT2AF2ALDH1A1MAPT
SCHEMBL304365 0.81 ALDH1A1 (0.40) MEN1KMT2AALDH1A1
SCHEMBL304341 0.79 PARP10 (0.41) PARP10PLA2G10PLA2G2ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160151322-A1 METALLO-B-LACTAMASE INHIBITORS MEIJI SEIKA KAISHA (JP) 2016-06-02 US disclosed
US-9260375-B2 Metallo-β-lactamase inhibitors MEIJI SEIKA KAISHA, LTD. (JP) 2016-02-16 US disclosed
US-20120071457-A1 METALLO-BETA-LACTAMASE INHIBITORS CHIKAUCHI KEN (JP) 2012-03-22 US disclosed
US-8093294-B2 Bacterial infections; effective for recovering the activities of beta-lactam antibiotics; 2-ethyl-3-methylmaleic acid dimethyl ester; maleic acid derivatives and/or dihydrofuranyl derivatives MEIJI SEIKA KAISHA, LTD. (JP) 2012-01-10 US disclosed
EP-1941873-A1 METALLO-BETA-LACTAMASE INHIBITOR MEIJI SEIKA KAISHA LTD. (JP) 2008-07-09 EP disclosed
US-20080090825-A1 Metallo-beta-lactamase inhibitors MEIJI SEIKA KAISHA, LTD. (JP) 2008-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080090825-A1 Metallo-beta-lactamase inhibitors ME1, MGAM, GAA PARP10 3704/4885PLA2G10 2962/4885PLA2G2A 3003/4885
US-20120071457-A1 METALLO-BETA-LACTAMASE INHIBITORS ME1, MGAM, GAA PARP10 3704/4885PLA2G10 2962/4885PLA2G2A 3003/4885
US-20160151322-A1 METALLO-B-LACTAMASE INHIBITORS ME1, MGAM, MANBA PARP10 3631/4885PLA2G10 2940/4885PLA2G2A 2871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.