SCHEMBL30437871

SCHEMBL30437871

Nc1ccc2ccc(-n3cccn3)cc2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 4/20 0.55
NOTUM Q6P988 1/20 0.46
BACE1 P56817 2/20 0.43
NCF1 P14598 2/20 0.43
NOS2 P35228 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
MPO P05164 2/20 0.41
LRRK2 Q5S007 1/20 0.39
LCK P06239 1/20 0.39
KIT P10721 1/20 0.39
SRC P12931 1/20 0.39
KDR P35968 1/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.38
PDK2 Q15119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30437851 0.79 CHRNA7 (0.49) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL20641982 0.78 NLRP3 (0.62) NLRP3NOTUMBACE1KDM4EALDH1A1
SCHEMBL30437703 0.78 NLRP3 (0.62) NLRP3NOTUMBACE1KDM4EALDH1A1
SCHEMBL20651722 0.75 NLRP3 (0.76) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL3665773 0.74 NOTUM (0.53) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL5337022 0.74 NOTUM (0.53) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL20641899 0.74 NLRP3 (0.71) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL3974447 0.73 HRH3 (0.53) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL29614982 0.73 NOTUM (0.52) NLRP3NOTUMKDM4EALDH1A1MAPK1
SCHEMBL17743393 0.73 NOTUM (0.52) NLRP3NOTUMKDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111793060-B NLRP3 modulators 先天肿瘤免疫公司 2023-06-06 CN disclosed