SCHEMBL3044737

SCHEMBL3044737

Cc1cc2nc[nH]c2cc1-c1ccc(CN(CCCC2CCCCC2)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 3/20 0.33
BRS3 P32247 1/20 0.33
QPCT Q16769 2/20 0.32
EPHX1 P07099 1/20 0.32
STAT3 P40763 1/20 0.32
AGTR1 P30556 1/20 0.31
HPGD P15428 1/20 0.31
HSD11B1 P28845 1/20 0.31
SLC2A1 P11166 1/20 0.31
TDP1 Q9NUW8 2/20 0.31
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
GSK3A P49840 1/20 0.31
MELK Q14680 1/20 0.30
OXTR P30559 1/20 0.30
AVPR1A P37288 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30
MAP4K1 Q92918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050687 0.95 HTR5A (0.34) HTR5ABRS3QPCTEPHX1STAT3
SCHEMBL3042077 0.92 QPCT (0.34) HTR5ABRS3QPCTEPHX1STAT3
SCHEMBL3044505 0.88 HTR5A (0.35) HTR5AEPHX1STAT3HSD11B1SLC2A1
SCHEMBL3047806 0.85 CDK1 (0.35) HTR5ABRS3EPHX1STAT3AGTR1
SCHEMBL3051515 0.83 HTT (0.37) BRS3QPCTAGTR1
SCHEMBL3046204 0.82 HTR5A (0.36) HTR5ABRS3EPHX1STAT3HSD11B1
SCHEMBL3048447 0.82 CNR2 (0.36) HTR5ABRS3AGTR1
SCHEMBL3054803 0.80 HTR5A (0.34) HTR5ABRS3AGTR1SLC2A1
Trifluoroacetic Acid SCHEMBL3044733 0.78 HTR5A (0.40) HTR5ABRS3EPHX1SLC2A1
SCHEMBL3041961 0.77 QPCT (0.33) QPCTOXTRAVPR1AMAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS OPRL1, OPRM1, OPRK1 HTR5A 190/4885BRS3 168/4885QPCT 1796/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.