SCHEMBL3048447

SCHEMBL3048447

Cc1nc2nc[nH]c2cc1-c1ccc(CN(CCC2CCCCC2)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.36
CNR1 P21554 1/20 0.36
HTR5A P47898 4/20 0.33
ABHD6 Q9BV23 1/20 0.33
BRS3 P32247 1/20 0.32
BCHE P06276 3/20 0.31
ACHE P22303 3/20 0.31
GUCY1B2 O75343 1/20 0.31
GUCY1A2 P33402 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
CSF1R P07333 1/20 0.31
ACVR1 Q04771 1/20 0.31
CCNB2 O95067 2/20 0.30
CDK1 P06493 2/20 0.30
CCNB1 P14635 2/20 0.30
CCNA2 P20248 2/20 0.30
CDK2 P24941 2/20 0.30
CCNA1 P78396 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050687 0.86 HTR5A (0.34) HTR5ABRS3BCHEACHEAGTR1
SCHEMBL3054803 0.84 HTR5A (0.34) HTR5ABRS3BCHEACHEAGTR1
SCHEMBL3047806 0.83 CDK1 (0.35) HTR5ABRS3BCHEACHECDK1
SCHEMBL3044737 0.82 HTR5A (0.33) HTR5ABRS3AGTR1
SCHEMBL3046204 0.81 HTR5A (0.36) HTR5ABRS3BCHEACHEHTR1A
SCHEMBL3042077 0.79 QPCT (0.34) HTR5ABRS3CDK1AGTR1
SCHEMBL3047275 0.79 CNR1 (0.31) CNR2CNR1ALOX5APFEN1
Trifluoroacetic Acid SCHEMBL3048446 0.78 HTR5A (0.41) CNR2CNR1HTR5AABHD6BRS3
SCHEMBL3044505 0.77 HTR5A (0.35) HTR5AHTR1ADRD2DRD4HTR1D
SCHEMBL3046358 0.77 PKM (0.32) HTR5ABRS3CSF1RAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS OPRL1, OPRM1, OPRK1 CNR2 25/4885CNR1 19/4885HTR5A 190/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.