SCHEMBL30452501

SCHEMBL30452501

Nc1cccn(-c2ccc(F)cn2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 5/20 0.47
MAPT P10636 6/20 0.38
GRM5 P41594 4/20 0.34
GRM3 Q14832 1/20 0.33
DHFR P00374 1/20 0.33
SLC27A1 Q6PCB7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20689567 1.00 TYK2 (0.47) TYK2MAPTGRM5GRM3DHFR
SCHEMBL23753623 0.81 NOS3 (0.39) TYK2GRM5DHFR
SCHEMBL16812410 0.81 ALDH1A1 (0.37) TYK2MAPTGRM5
SCHEMBL30174271 0.80 TYK2 (0.56) TYK2SLC27A1
SCHEMBL31572570 0.79 TYK2 (0.32) TYK2MAPT
SCHEMBL20689381 0.78 TYK2 (0.40) TYK2MAPTGRM5DHFR
SCHEMBL20687706 0.78 TYK2 (0.54) TYK2
SCHEMBL31563759 0.78 MAPT (0.33) TYK2MAPT
SCHEMBL25208803 0.78 TYK2 (0.47) TYK2MAPTSLC27A1
SCHEMBL18161077 0.78 GPR119 (0.34) TYK2DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916207-A Five-membered and six-membered heterocyclic compounds and application thereof as protein receptor kinase inhibitors 轶诺(浙江)药业有限公司 2023-04-04 CN disclosed