SCHEMBL30453653

SCHEMBL30453653

CN1CCC(NC(=O)c2ccc(-c3cnc(N)c(OCc4cccc(F)c4C(F)(F)F)n3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATR Q13535 5/20 0.54
PTK2 Q05397 6/20 0.47
SLC6A5 Q9Y345 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
KCNH2 Q12809 1/20 0.42
CHEK2 O96017 1/20 0.42
MET P08581 1/20 0.42
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41
HDAC1 Q13547 1/20 0.41
CSF1R P07333 1/20 0.41
AXL P30530 1/20 0.40
MERTK Q12866 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL487938 1.00 ATR (0.54) ATRPTK2SLC6A5HDAC4HDAC6
SCHEMBL488735 0.85 MET (0.49) ATRPTK2SLC6A5HDAC4HDAC6
SCHEMBL30454046 0.85 MET (0.49) ATRPTK2SLC6A5HDAC4HDAC6
SCHEMBL488626 0.85 KCNH2 (0.56) ATRKCNH2
SCHEMBL30454874 0.85 KCNH2 (0.56) ATRKCNH2
SCHEMBL30452854 0.82 CD274 (0.50) ATR
SCHEMBL488001 0.82 CD274 (0.50) ATR
SCHEMBL30453567 0.81 ATR (0.55) ATRSLC6A5HDAC4HDAC6CHEK2
SCHEMBL488430 0.81 ATR (0.55) ATRSLC6A5HDAC4HDAC6CHEK2
SCHEMBL488522 0.81 MAP4K4 (0.43) ATRKCNH2CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed