SCHEMBL30457411

SCHEMBL30457411

C[C@@H]1CN(c2nccc(CN)n2)C[C@H](C)N1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 3/20 0.43
GHSR Q92847 1/20 0.37
EIF2AK4 Q9P2K8 1/20 0.36
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 2/20 0.35
BCL6 P41182 3/20 0.35
NCOR2 Q9Y618 1/20 0.35
ATR Q13535 1/20 0.34
ATRIP Q8WXE1 1/20 0.34
SCN9A Q15858 1/20 0.34
KHK P50053 1/20 0.32
ACHE P22303 2/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
SORD Q00796 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25240554 1.00 PTPN11 (0.43) PTPN11GHSREIF2AK4ROCK2ROCK1
SCHEMBL3533723 0.80 PTPN11 (0.48) PTPN11GHSREIF2AK4ROCK2ROCK1
SCHEMBL3533726 0.80 PTPN11 (0.48) PTPN11GHSREIF2AK4ROCK2ROCK1
SCHEMBL25238416 0.77 CHRM2 (0.38) SORD
SCHEMBL25234344 0.75 PTPN11 (0.38) PTPN11GHSREIF2AK4HDAC1
SCHEMBL31421576 0.74 ACHE (0.43) ACHESORDPIK3CAMTOR
SCHEMBL25236876 0.73 EIF2AK4 (0.43) EIF2AK4SORD
SCHEMBL30457520 0.73 EIF2AK4 (0.43) EIF2AK4SORD
SCHEMBL25280102 0.73 CTSS (0.42) PTPN11GHSRROCK2ROCK1
SCHEMBL29631769 0.73 KDM4E (0.44) PTPN11GHSRSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023110843-A1 HETEROBICYCLIC DERIVATIVES AS ITK INHIBITORS ALMIRALL, S.A. (ES) 2023-06-22 WO disclosed