SCHEMBL30458225

SCHEMBL30458225

CC(OC(N)=O)c1ccc(OCCOCCOc2ccc(C(C)OC(N)=O)nc2)cn1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
RARB P10826 1/20 0.35
PARP10 Q53GL7 2/20 0.35
CACNA1I Q9P0X4 2/20 0.34
CACNA1G O43497 1/20 0.34
CACNA1H O95180 1/20 0.34
CNR2 P34972 1/20 0.34
KCNH2 Q12809 1/20 0.34
CYP4F2 P78329 2/20 0.34
CYP4A11 Q02928 2/20 0.34
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15764197 0.78 PDE3B (0.39) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL22604308 0.77 NCF1 (0.38) KDM4EMAPK1
SCHEMBL22604304 0.77 NCF1 (0.38) KDM4EMAPK1
SCHEMBL22587373 0.76 ESR1 (0.45)
SCHEMBL27774508 0.76 MAPT (0.43) MAPT
SCHEMBL27166286 0.75 PPARG (0.39) KDM4ERARBPARP10MAPT
SCHEMBL22587389 0.75 KDM4E (0.40) KDM4EMAPK1MAPT
SCHEMBL4204388 0.75 APLNR (0.50) MAPK1
SCHEMBL28172147 0.75 KMO (0.40) KDM4EMAPK1
SCHEMBL22604307 0.73 CACNA1I (0.47) CACNA1ICACNA1GCACNA1HCNR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825666-B Dimeric or multimeric forms of mutant IDH inhibitors 上海仕谱生物科技有限公司 2024-03-08 CN disclosed
CN-114127060-B Dimeric or multimeric forms of mutant IDH inhibitors 上海仕谱生物科技有限公司 2023-06-13 CN disclosed