SCHEMBL30480705

SCHEMBL30480705

O=C(CBr)c1cc2[nH]ncc2cc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.46
NOS1 P29475 3/20 0.45
METAP2 P50579 2/20 0.45
DYRK1A Q13627 2/20 0.45
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CSNK2A1 P68400 1/20 0.41
CTNNB1 P35222 5/20 0.40
WNT3A P56704 5/20 0.40
CASP6 P55212 1/20 0.40
CHEK1 O14757 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
HTT P42858 1/20 0.38
FGFR1 P11362 1/20 0.37
FGFR2 P21802 1/20 0.37
FGFR3 P22607 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL616074 1.00 AXL (0.46) AXLNOS1METAP2DYRK1ANPC1
SCHEMBL22446038 0.82 CASP6 (0.54) AXLNOS1METAP2DYRK1ANPC1
SCHEMBL617024 0.81 AXL (0.53) AXLNOS1METAP2DYRK1ANPC1
SCHEMBL18554980 0.77 AXL (0.56) AXLNOS1METAP2DYRK1ANPC1
SCHEMBL30286390 0.77 AXL (0.56) AXLNOS1METAP2DYRK1ANPC1
SCHEMBL2926007 0.76 PTPN1 (0.51) NOS1METAP2DYRK1ACTNNB1WNT3A
SCHEMBL616794 0.76 NOS1 (0.44) NOS1CTNNB1WNT3ACHEK1MEN1
SCHEMBL15059952 0.73 CTNNB1 (0.67) NOS1METAP2DYRK1ANPC1RAB9A
SCHEMBL616185 0.73 AXL (0.51) AXLNOS1METAP2DYRK1ANPC1
SCHEMBL26322070 0.72 ALDH1A1 (0.46) AXLNPC1RAB9ACTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107973809-B Macrocyclic compounds as factor XIA inhibitors 百时美施贵宝公司 2023-06-30 CN disclosed