SCHEMBL3048579

SCHEMBL3048579

Nc1c(-c2ccc(CO)cc2)cc(Br)c2c1C(=O)NC2=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.43
WEE1 P30291 5/20 0.43
HPGD P15428 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
PRKAB2 O43741 3/20 0.32
PRKAG1 P54619 3/20 0.32
PRKAA2 P54646 3/20 0.32
PRKAA1 Q13131 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3048914 0.87 WEE1 (0.51) CHEK1WEE1HPGDMMP2MMP9
SCHEMBL3046283 0.82 MAPT (0.40) CHEK1WEE1GSK3B
SCHEMBL3044714 0.78 CHEK1 (0.45) CHEK1WEE1GSK3BBRD4
SCHEMBL1425210 0.70 GAA (0.37) CHEK1WEE1CA1CA2CA9
SCHEMBL3037404 0.69 TDP2 (0.37) HPGDIKBKB
SCHEMBL3040023 0.69 CHEK1 (0.42) CHEK1WEE1HPGDGSK3BIKBKB
SCHEMBL3044668 0.67 WEE1 (0.46) CHEK1WEE1GSK3B
SCHEMBL3038080 0.66 CA1 (0.39) CHEK1WEE1CA1CA2CA7
SCHEMBL30440457 0.64 CSNK2A2 (0.54) CHEK1WEE1HPGDCA12CA1
SCHEMBL28133857 0.62 PPOX (0.50) HPGDGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745641-B2 Nitrogen-containing heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-06-29 US disclosed
US-20090054407-A1 Nitrogen-containing heterocyclic compound KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-02-26 US disclosed
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054407-A1 Nitrogen-containing heterocyclic compound NR4A1, NR5A2, PRMT8 CHEK1 3306/4885WEE1 965/4885HPGD 2485/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.