SCHEMBL30487

SCHEMBL30487

Cc1cc(F)c(C(=O)Nc2nc3ccc(O)cc3s2)c(Cl)c1O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 8/20 0.72
HSD17B2 P37059 7/20 0.72
CYP3A4 P08684 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2B6 P20813 1/20 0.62
CYP2C19 P33261 1/20 0.62
DYRK1A Q13627 2/20 0.55
NPC1 O15118 5/20 0.49
RAB9A P51151 5/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
HSD17B10 Q99714 1/20 0.48
LRRK2 Q5S007 1/20 0.48
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30432 0.84 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29964 0.77 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29710 0.76 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL13329428 0.75 DYRK1A (0.62) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29886 0.74 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29870 0.74 HSD17B1 (0.75) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL544349 0.73 DYRK1A (0.75) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL12199323 0.73 HSD17B1 (0.76) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL13329360 0.73 HSD17B1 (0.74) HSD17B1HSD17B2DYRK1ANPC1RAB9A
SCHEMBL12199347 0.73 HSD17B1 (0.76) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed