SCHEMBL30487408

SCHEMBL30487408

N#Cc1cc(Br)cc(F)c1N

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.42
ADRB1 P08588 1/20 0.42
KHK P50053 1/20 0.39
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
TRPV4 Q9HBA0 3/20 0.36
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
XDH P47989 1/20 0.33
GPR35 Q9HC97 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
EGLN2 Q96KS0 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3230060 1.00 ADRB2 (0.42) ADRB2ADRB1KHKCYP11B1CYP11B2
SCHEMBL9478745 0.84 XDH (0.37) ADRB2KHKXDHGPR35MAOA
SCHEMBL31020001 0.82 KHK (0.40) ADRB2ADRB1KHKCYP11B1CYP11B2
SCHEMBL29560065 0.78 TRPV4 (0.39) KHKCYP11B1CYP11B2TRPV4GPR35
SCHEMBL144243 0.78 ADRB2 (0.43) ADRB2CA1CA2CA9XDH
SCHEMBL2652439 0.78 ADRB2 (0.44) ADRB2ADRB1KHKCYP11B1CYP11B2
SCHEMBL504867 0.78 TRPV4 (0.39) KHKCYP11B1CYP11B2TRPV4GPR35
SCHEMBL18343829 0.78 XDH (0.34) ADRB2XDHGPR35MAOAMAOB
SCHEMBL29582221 0.78 ADRB2 (0.43) ADRB2CA1CA2CA9XDH
SCHEMBL58096 0.77 HDAC1 (0.44) ADRB2CA1CA2CA9HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125935-A1 BENZOPYRIDINE DERIVATIVE REGULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2023-07-06 WO disclosed