SCHEMBL30489012

SCHEMBL30489012

Nc1ccc2[nH]c(-c3ccc(N4CCNCC4)cc3)nc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.52
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
RXFP1 Q9HBX9 2/20 0.51
CACNA1B Q00975 1/20 0.51
APBA1 Q02410 1/20 0.51
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 5/20 0.50
MAPT P10636 5/20 0.50
SMN1; SMN2 Q16637 5/20 0.50
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
GLA P06280 3/20 0.50
GFER P55789 3/20 0.50
GAA P10253 3/20 0.50
RECQL P46063 2/20 0.50
HPGD P15428 4/20 0.48
HSD17B10 Q99714 3/20 0.48
POLB P06746 2/20 0.48
NFKB1 P19838 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25274071 1.00 PARP1 (0.52) PARP1MEN1KMT2ARXFP1CACNA1B
SCHEMBL1663221 0.87 PARP1 (0.52) PARP1MEN1KMT2ARXFP1CACNA1B
SCHEMBL31289499 0.86 DGAT1 (0.58) PARP1MEN1KMT2ARXFP1CACNA1B
SCHEMBL10325591 0.84 HTR3E (0.51) PARP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL30533210 0.82 MEN1 (0.73) MEN1KMT2ARXFP1CACNA1BAPBA1
SCHEMBL1655753 0.82 MEN1 (0.73) MEN1KMT2ARXFP1CACNA1BAPBA1
SCHEMBL14669422 0.81 PARP1 (0.44) PARP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL532061 0.81 ACHE (0.68) PARP1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL19137933 0.81 RHEB (0.58) PARP1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL159873 0.80 ALDH1A1 (0.74) MEN1KMT2ARXFP1CACNA1BAPBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023110765-A1 BENZIMIDAZOLE DERIVATIVES FOR THE TREATMENT AND PROPHYLAXIS OF INFECTIOUS DISEASES EBERHARD KARLS UNIVERSITAET TUEBINGEN MEDIZINISCHE FAKULTAET (DE) 2023-06-22 WO disclosed