Taranabant

Taranabant

SCHEMBL304925

C[C@H](NC(=O)C(C)(C)Oc1ccc(C(F)(F)F)cn1)[C@@H](Cc1ccc(Cl)cc1)c1cccc(C#N)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CNR1

The experimentally established mechanism targets of Taranabant. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR1 known ✓ P21554 20/20 1.00
CNR2 P34972 9/20 1.00
CYP2D6 P10635 1/20 1.00
CYP2C9 P11712 1/20 1.00
KCNH2 Q12809 1/20 1.00
CYP3A4 P08684 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Taranabant SCHEMBL17565778 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
Taranabant SCHEMBL13253304 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
Taranabant SCHEMBL501972 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
Taranabant SCHEMBL4024243 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
Taranabant SCHEMBL29434856 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
Taranabant SCHEMBL13253294 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3474367 0.95 CNR1 (0.90) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3474366 0.95 CNR1 (0.90) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3475455 0.93 CNR1 (0.87) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL16357820 0.93 CNR1 (0.87) CNR1CNR2CYP2D6CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 702 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US claimed
US-20250352559-A1 Transdermal Delivery Composition for Delivery of at least one Glucose Controlling Agent, and Method of Delivering at least one Glucose Controlling Agent SKINVISIBLE PHARMACEUTICALS INC (US) 2025-11-20 US claimed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4486336-A2 CB1 LIGAND CONJUGATED COMPOUNDS AND USES THEREOF Adarx Pharmaceuticals, Inc. (US) 2025-01-08 EP claimed
US-20240408059-A1 METHOD OF TREATING ADDICTION ANEBULO PHARMACEUTICALS, INC. 2024-12-12 US claimed
WO-2024107445-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES, INC. (US) 2024-05-23 WO claimed
US-20230330111-A1 ACTIVE AGENT COMBINATION FOR TREATMENT OF CANCER Helmholtz Zentrum München - Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) (DE) 2023-10-19 US claimed
WO-2023168296-A2 CB1 LIGAND CONJUGATED COMPOUNDS AND USES THEREOF ADARX PHARMACEUTICALS, INC. (US) 2023-09-07 WO claimed
EP-4203944-A1 ACTIVE AGENT COMBINATION FOR TREATMENT OF CANCER Helmholtz Zentrum München Deutsches Forschungszentrum für Gesundheit und Umwelt GmbH (DE) 2023-07-05 EP claimed
WO-2022198259-A1 TREATMENT METHODS FOR PULMONARY ARTERIAL HYPERTENSION THE HEART RESEARCH INSTITUTE LTD (AU) 2022-09-29 WO claimed
WO-2022043490-A1 ACTIVE AGENT COMBINATION FOR TREATMENT OF CANCER Helmholtz Zentrum München - Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) (DE) 2022-03-03 WO claimed
EP-2739262-B1 USE OF A CB1 RECEPTOR ANTAGONIST AS A WHITENING AND/OR ANTI-BROWNING AGENT FOR KERATIN MATERIAL OREAL (FR) 2017-09-27 EP claimed
US-9662320-B2 Antagonists of the cannabinoid receptor CB1 for use in the treatment of diseases associated with neuronal dendritic abnormalities UNIVERSITAT POMPEU FABRA (ES) 2017-05-30 US claimed
US-20160067235-A1 Antagonists of the Cannabinoid Receptor CB1 for Use in the Treatment of Diseases Associated with Neuronal Dendritic Abnormalities UNIVERSITAT POMPEU FABRA (ES) 2016-03-10 US claimed
EP-2739262-A2 USE OF A CB1 RECEPTOR ANTAGONIST AS A WHITENING AND/OR ANTI-BROWNING AGENT FOR KERATIN MATERIAL L'OREAL (FR) 2014-06-11 EP claimed
US-8715648-B2 Method for treating obesity with anti-obesity formulations and omega 3 fatty acids for the reduction of body weight in cardiovascular disease patients (CVD) and diabetics PIVOTAL THERAPEUTICS INC. (CA) 2014-05-06 US claimed
WO-2013021129-A2 USE OF A CB1 RECEPTOR ANTAGONIST AS A WHITENING AND/OR ANTI-BROWNING AGENT FOR KERATIN MATERIAL L'OREAL (FR) 2013-02-14 WO claimed
US-20090306037-A1 Combination of a Dipeptidyl Peptidase-IV Inhibitor and a Cannabinoid CB1 Receptor Antagonist for the Treatment of Diabetes and Obesity MERCK & CO., INC. (US) 2009-12-10 US claimed
US-20060270650-A1 Combination therapy for the treatment of obesity MACNEIL TANYA 2006-11-30 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240408059-A1 METHOD OF TREATING ADDICTION CNR2, CNR1, OPRM1 CNR1 2/4885CNR2 1/4885CYP2D6 533/4885
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES PDE9A, PDE3A, PDE2A CNR1 221/4885CNR2 204/4885CYP2D6 1028/4885
US-20230330111-A1 ACTIVE AGENT COMBINATION FOR TREATMENT OF CANCER GLS2, AGK, GLS CNR1 3466/4885CNR2 3282/4885CYP2D6 2211/4885
US-20250352559-A1 Transdermal Delivery Composition for Delivery of at least one Glucose Controlling Agent, and Method of Delivering at least one Glucose Controlling Agent SLC2A1, SLC2A4, SLC2A8 CNR1 2558/4885CNR2 3030/4885CYP2D6 1106/4885
US-20090306037-A1 Combination of a Dipeptidyl Peptidase-IV Inhibitor and a Cannabinoid CB1 Receptor Antagonist for the Treatment of Diabetes and Obesity DPP4, DPP3, DPP7 CNR1 6/4885CNR2 10/4885CYP2D6 831/4885
US-20160067235-A1 Antagonists of the Cannabinoid Receptor CB1 for Use in the Treatment of Diseases Associated with Neuronal Dendritic Abnormalities CNR1, CNR2, DBN1 CNR1 1/4885CNR2 2/4885CYP2D6 4659/4885
US-20060270650-A1 Combination therapy for the treatment of obesity GPR119, GANC, GANAB CNR1 385/4885CNR2 281/4885CYP2D6 4112/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.