SCHEMBL30513601

SCHEMBL30513601

O=c1c(NCc2ccccn2)c(Nc2ccc(Cl)c(Cl)c2)c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.56
GLA P06280 1/20 0.56
HTT P42858 1/20 0.56
CHEK1 O14757 2/20 0.54
MAP4K4 O95819 2/20 0.54
CHEK2 O96017 2/20 0.54
PRKACA P17612 2/20 0.54
RPS6KB1 P23443 2/20 0.54
AKT1 P31749 2/20 0.54
GSK3A P49840 2/20 0.54
GSK3B P49841 2/20 0.54
RPS6KA3 P51812 2/20 0.54
NEK4 P51957 2/20 0.54
CSNK1G2 P78368 2/20 0.54
PRKCD Q05655 2/20 0.54
PRKAA1 Q13131 2/20 0.54
PRKG2 Q13237 2/20 0.54
ROCK1 Q13464 2/20 0.54
PRKG1 Q13976 2/20 0.54
PKN2 Q16513 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28641831 1.00 MAPT (0.56) MAPTGLAHTTCHEK1MAP4K4
SCHEMBL28633070 0.86 CHEK1 (0.58) CHEK1MAP4K4CHEK2PRKACARPS6KB1
SCHEMBL28637102 0.83 MAOA (0.63) CHEK1MAP4K4CHEK2PRKACARPS6KB1
SCHEMBL28653147 0.81 PIK3CA (0.51) KMT2AALDH1A1MAOAMAOBNPC1
SCHEMBL30513615 0.81 PIK3CA (0.51) KMT2AALDH1A1MAOAMAOBNPC1
SCHEMBL28635668 0.81 MAPKAPK2 (0.50) MAPTCHEK1MAP4K4CHEK2PRKACA
SCHEMBL28651333 0.81 CHEK1 (0.52) MAPTHTTCHEK1MAP4K4CHEK2
SCHEMBL28642296 0.81 CHEK2 (0.58) MAPTCHEK1MAP4K4CHEK2PRKACA
SCHEMBL28640083 0.81 KMT2A (0.53) MAPTCHEK1MAP4K4CHEK2PRKACA
SCHEMBL28925293 0.81 MAPKAPK2 (0.50) MAPTCHEK1MAP4K4CHEK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759549-B 3-substituted amino-4- ((substituted pyridinyl) amino) cyclobut-3-ene-1, 2-dione compounds 中国医学科学院药物研究所 2023-07-28 CN disclosed