SCHEMBL30516078

SCHEMBL30516078

O=Cc1ncc(-c2ncon2)cc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.41
KCNH2 Q12809 4/20 0.39
CNR1 P21554 1/20 0.36
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
S1PR1 P21453 5/20 0.34
S1PR3 Q99500 2/20 0.34
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
PTPN11 Q06124 1/20 0.32
KMO O15229 1/20 0.32
TOP1 P11387 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493936 0.77 KIF11 (0.45) KCNH2CNR1S1PR1S1PR3CHUK
SCHEMBL30516088 0.76 CNR1 (0.38) MAP4K4KCNH2CNR1CA12CA9
SCHEMBL30516067 0.75 HDAC4 (0.34) MAP4K4KCNH2CNR1S1PR1S1PR3
SCHEMBL24799621 0.68 IDH1 (0.40) KCNH2CNR1S1PR1S1PR3NPC1
SCHEMBL19836179 0.67 S1PR1 (0.41) KCNH2CNR1S1PR1S1PR3MAPT
SCHEMBL27951856 0.67 TOP1 (0.48) TOP1
SCHEMBL30516110 0.67 PPARA (0.41) KMO
SCHEMBL29045046 0.67 PPARA (0.41) KMO
SCHEMBL28601834 0.66 PTGS2 (0.48) S1PR1S1PR3ALDH1A1MAPTRAB9A
SCHEMBL472486 0.66 GSK3B (0.46) KCNH2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN claimed
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN disclosed