SCHEMBL30516088

SCHEMBL30516088

O=Cc1cc(-c2ccc(C(F)(F)F)cc2)cc(-c2ncon2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.38
KCNH2 Q12809 1/20 0.38
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
KIF11 P52732 5/20 0.36
P2RY14 Q15391 2/20 0.35
S1PR1 P21453 3/20 0.34
DHODH Q02127 1/20 0.34
S1PR3 Q99500 2/20 0.34
HDAC1 Q13547 1/20 0.34
MCHR1 Q99705 1/20 0.34
MAP4K4 O95819 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
HCRTR1 O43613 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493936 0.80 KIF11 (0.45) CNR1KCNH2KIF11S1PR1S1PR3
SCHEMBL30516078 0.76 MAP4K4 (0.41) CNR1KCNH2CA12CA9S1PR1
SCHEMBL6851712 0.73 BRD4 (0.42) PPARA
SCHEMBL19836179 0.73 S1PR1 (0.41) CNR1KCNH2S1PR1S1PR3RXRA
SCHEMBL30516067 0.73 HDAC4 (0.34) CNR1KCNH2S1PR1S1PR3MAP4K4
SCHEMBL1175073 0.71 BRD4 (0.48) CA12CA9PPARACA1CA2
SCHEMBL18002017 0.71 MAPT (0.42) KIF11CA1CA2
SCHEMBL29955861 0.71 BRD4 (0.48) CA12CA9PPARACA1CA2
SCHEMBL28601834 0.71 PTGS2 (0.48) S1PR1S1PR3CA1CA2CYP3A4
SCHEMBL24386409 0.70 GPR119 (0.37) CNR1KCNH2S1PR1S1PR3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN claimed
CN-116514790-A Tri-aromatic heterocyclic piperazine small molecular organic compound targeting STAT3 and application thereof 华东师范大学 2023-08-01 CN disclosed