SCHEMBL30572694

SCHEMBL30572694

[2H]c1cc(-c2cc3c(N4CCNCC4)ccnn3c2)cnc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.45
RIOK2 Q9BVS4 4/20 0.40
NCF1 P14598 2/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
KIT P10721 3/20 0.38
ACVR1 Q04771 2/20 0.38
TGFBR1 P36897 1/20 0.38
HTR3A P46098 2/20 0.37
HTR6 P50406 2/20 0.37
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR7 P34969 1/20 0.37
HTR2B P41595 1/20 0.37
MTOR P42345 2/20 0.36
RPTOR Q8N122 1/20 0.36
MLST8 Q9BVC4 1/20 0.36
ADRB1 P08588 2/20 0.36
HTR3E A5X5Y0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30572725 0.91 RET (0.49) RETRIOK2NCF1CHRNB2CHRNA4
SCHEMBL19462890 0.73 RET (0.45) RETNCF1KITACVR1TGFBR1
SCHEMBL19459259 0.69 LIPG (0.43) RETNCF1KITACVR1TGFBR1
SCHEMBL19481688 0.69 RET (0.54) RET
SCHEMBL19458933 0.69 NCF1 (0.48) RETNCF1HTR3AHTR6HTR2A
SCHEMBL19482443 0.68 RET (0.41) RETNCF1KITACVR1TGFBR1
SCHEMBL30333672 0.68 CYP1A2 (0.53) RIOK2HTR2CCYP2C19PIK3CDPIK3CA
SCHEMBL30333558 0.68 CYP1A2 (0.64) CYP2C19PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL21679774 0.68 KHK (0.43) RETKITACVR1TGFBR1BMPR1B
Hydrochloric Acid SCHEMBL19459005 0.68 NCF1 (0.47) RETNCF1HTR3AHTR6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023165581-A1 PYRIDINE DERIVATIVE AND USE THEREOF 四川汇宇制药股份有限公司 2023-09-07 WO disclosed