SCHEMBL30585261

SCHEMBL30585261

COc1ccc(CN2CCN(CC(=O)Nc3ccc(OC)nc3)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.61
KDM4E B2RXH2 3/20 0.61
OGA O60502 1/20 0.57
REV1 Q9UBZ9 1/20 0.56
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
MAPT P10636 2/20 0.56
KCNA5 P22460 2/20 0.55
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
GFER P55789 1/20 0.54
GAA P10253 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29078372 1.00 ALDH1A1 (0.61) ALDH1A1KDM4EOGAREV1MEN1
SCHEMBL29078382 0.90 MEN1 (0.65) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL30585251 0.90 MEN1 (0.65) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL29078394 0.87 MEN1 (0.60) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL29078389 0.80 MYD88 (0.60) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL29078402 0.79 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL30585253 0.77 TSHR (0.47) ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL22516942 0.76 LSS (0.65) ALDH1A1KDM4EMEN1KMT2ACYP3A4
SCHEMBL12244095 0.76 ACHE (0.58) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL30585252 0.76 OGA (0.51) ALDH1A1KDM4EOGAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN claimed
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN disclosed